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[(4-fluorophenyl)methyl]({[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(prop-2-en-1-yl)amine
2-benzyl-3-methyl-4-(1-methyl-1H-imidazol-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-{1-[2-(2-butyl-5-chloro-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{1-[(dimethyl-1,3-thiazol-4-yl)methyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
8-(2-amino-6-methylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{[ethyl(oxolan-2-ylmethyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(cyclopropylmethyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-2-(methylamino)pyrimidine-5-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2-(2-methylphenyl)ethan-1-one
N-methyl-2-{2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}acetamide
1-(3-chlorothiophene-2-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azepan-2-yl}methanol
1-cyclobutanecarbonyl-4-(2-methylphenoxy)piperidine
7-(2-amino-6-methoxypyrimidin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(3-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}phenyl)acetamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-(2-ethoxypyridin-3-yl)-4-methoxypyrimidine
5-oxo-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-3-carboxylic acid
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
N-methyl-N-(oxan-2-ylmethyl)-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
4-[5-(1-hydroxypropyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]-1-methyl-1,2-dihydroquinolin-2-one
3-ethyl-5-methyl-4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,2-oxazole
{4-[(4-chlorophenyl)methyl]-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}methanol
dimethyl[3-(2-{1-[4-(propan-2-yl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-4-methoxy-3,5-dimethylpyridine
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-yl]acetamide
1-(cyclohexylmethyl)-3-methyl-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-(2-{2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}propyl)-1H-1,2,4-triazole
N-(2,4-dimethylphenyl)-2-{[1-(morpholin-4-ylmethyl)cyclopentyl]amino}acetamide
(2S,4R)-4-[4-({[(2,5-dimethylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-[(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]acetic acid
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}-1H-pyrazole-4-carboxamide
5-(3-chlorophenyl)-N-[2-(piperidin-1-yl)ethyl]-1,2,4-triazin-3-amine
2-[(methylcarbamoyl)methyl]-N-[4-(morpholin-4-ylmethyl)phenyl]-3-oxopiperazine-1-carboxamide
4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2-methyl-1,3-thiazole
2-(cyclohex-1-en-1-yl)-N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(thiophene-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-methoxy-N,4-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
3-(2,1,3-benzothiadiazol-4-yl)-1-methyl-1-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]urea
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]propanamide
N-[(3-chlorophenyl)methyl]-3-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}propanamide
N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-1H-indazole-3-carboxamide
13-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
(1S,5R)-6-(2,3-dihydro-1H-indene-5-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(furan-2-yl)ethane-1,2-dione