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1-methyl-3-{5-[(4-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-(pyrimidin-4-ylmethyl)urea
5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-methylpropan-1-one
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]propan-1-one
8-[(3-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(oxan-4-yl)piperidine
1-[4-(4-fluorophenoxy)piperidin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
(2E)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-3-(thiophen-2-yl)prop-2-enamide
4-[7-(oxolane-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
N-methyl-3-(2-methylphenyl)-3-phenyl-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
5-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-2-(3,5-dichlorophenyl)pyrimidin-4-ol
5-(hydroxymethyl)-2-methyl-4-({2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)pyridin-3-ol
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)acetamide
N-(2,2-difluoroethyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonyl)morpholine
6-{4-[1-(dimethylamino)ethyl]phenyl}pyridin-3-ol
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,2-dihydrophthalazin-1-one
N-cyclopropyl-2-[4-(2-methylphenoxy)piperidin-1-yl]pyridine-4-carboxamide
{2-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]phenyl}methanol
2-(2-hydroxyethyl)-6-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
3-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
3-[1-butyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
1-ethyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-ethyl-N-[(2-methoxynaphthalen-1-yl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopropyl-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
3-{1-[3-(furan-2-yl)benzoyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4S)-N-ethyl-4-[2-(methylsulfanyl)acetamido]-1-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
methyl 2-{2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamido}-2-(3-methylphenyl)acetate
N-{3-[4-(thiomorpholin-4-yl)piperidin-1-yl]phenyl}-3-(trifluoromethyl)benzamide
1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidine-4-carbonitrile
7-(cyclobutylmethyl)-2-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[2-(phenylsulfanyl)acetyl]pyrrolidin-3-yl]acetamide
(2R,6R)-4-(1H-pyrrole-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[1-(pyridin-3-ylmethyl)piperidine-3-carbonyl]pyridine
1-(2-phenoxyethyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
N-[(4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}phenyl)methyl]methanesulfonamide
(benzylsulfamoyl)[(5-methoxy-1H-indol-2-yl)methyl]amine
3-({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(pyridin-4-ylmethyl)amino)propan-1-ol
6-[(oxolan-3-yl)amino]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
[4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-1,4-oxazepan-6-yl]methanol
1-ethyl-3-methyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]piperidine-3-carboxamide
1-[2-(5-methylfuran-2-yl)phenyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
methyl 1-[(3S,5S)-5-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 6-[(2-fluoro-5-methoxyphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N,N-dimethyl-3-(8-methylquinolin-5-yl)-1H-1,2,4-triazol-5-amine