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2-{2-[1-(4-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-(2-{[4-(dimethylamino)piperidin-1-yl]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-(propan-2-yloxy)propan-1-one
9-[(3-methylthiophen-2-yl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)azepan-2-one
8-[2-(3-chloro-4-fluorophenoxy)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N,1-dimethyl-2-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]imidazolidine-4-carboxamide
2-(3-fluoro-4-methylphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
N-[(1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}piperidin-4-yl)methyl]acetamide
5-(4-methylpyridin-3-yl)isoquinoline
N-(3-{[(2-propoxyethyl)carbamoyl]amino}phenyl)cyclopentanecarboxamide
2-benzyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(4aS,8aR)-6-[4-(aminomethyl)benzoyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-(2-methoxyethyl)-1-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-benzyl-3-{[1-(4,4,4-trifluorobutan-2-yl)piperidin-4-yl]oxy}benzamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(2,3,6-trifluorophenyl)methyl]piperidine
2-(2-ethyl-1H-imidazol-1-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}ethan-1-one
3-(1,2-oxazolidin-2-yl)-1-[2-(3-phenylpropyl)morpholin-4-yl]propan-1-one
N-(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
5-{2-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}-8-fluoroquinoline
1-[(3-fluorophenyl)methyl]-6-oxo-N-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-3-carboxamide
4-(1-methyl-1H-pyrazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{3-[3-(3-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
2-{9-[(2,4-dimethoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine-3-carboxamide
1-[(1-methylpiperidin-4-yl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
(1R,5R)-3-(3-chloro-2-methylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
6-cyclopentyl-1-methyl-N-[3-(pyridin-3-yloxy)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidin-2-yl)-5-(propan-2-yl)-1,2-oxazole
2-(3-methoxypropyl)-9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(carbamoylamino)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
3-[1-(6-methyl-4-oxo-4H-pyran-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
3-({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)-2-(thiophen-3-ylmethyl)propan-1-ol
4-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]-N-phenylpiperidine-1-carboxamide
2-chloro-4-(3-cyclopropyl-1-ethyl-1H-1,2,4-triazol-5-yl)phenol
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
2-methyl-6-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)pyrimidin-4-ol
1-{4-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]phenyl}imidazolidine-2,4-dione
1-(4-chloro-2-hydroxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
4-({2,4-dimethyl-5-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
2-amino-N-[2-(6-methoxynaphthalen-2-yl)phenyl]acetamide
N-methyl-6-(propane-1-sulfonyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
ethyl 4-{1-[(1R)-1-carbamoylethyl]-4-phenyl-1H-imidazol-5-yl}-1H-pyrazole-3-carboxylate
N-[(3-{[(2S,5R)-5-(morpholin-4-ylmethyl)oxolan-2-yl]methyl}phenyl)methyl]propanamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(5-fluoro-2-methyl-1H-indol-3-yl)acetamide
6-methyl-2-(oxan-4-yl)-5-[5-(1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine