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2-cyclooctyl-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
6-fluoro-2-oxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
(2R,3R,6R)-5-(3,4-difluorobenzoyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-butyl-3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(3-fluorophenyl)piperidine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methyl-1,3-benzoxazole-6-carboxamide
2-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
1-{3-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
6-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
7-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
ethyl 1-(1H-indazole-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyridin-4-yl)piperazine
N-[2-(phenylsulfanyl)ethyl]-N-(propan-2-yl)-1H-pyrrole-2-carboxamide
(3E)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]hept-3-enoic acid
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)acetamide
3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-7-methyl-1,2-dihydroquinolin-2-one
1-(1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-1-oxopropan-2-yl)pyrrolidin-2-one
4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-sulfonyl]-N-[(5-methylfuran-2-yl)methyl]benzamide
5,5-dimethyl-3-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1,3-oxazolidine-2,4-dione
4-[2-(4-fluorophenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]-4-(4-fluorophenyl)butane-1,4-dione
6-[(carbamoylmethyl)amino]-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]pyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)acetamide
3-(3-fluoro-4-phenylbenzoyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
2-[3-oxo-9-(3-phenoxypropanoyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2-(3-{[4-(4-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]methyl}phenoxy)acetamide
2-methyl-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
dimethyl(3-{2-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
(4aS,7aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methoxy-3-methyl-N-[1-(1,3-thiazol-5-yl)propan-2-yl]-1-benzofuran-2-carboxamide
(2S,4R)-N,N-diethyl-4-[2-(3-fluorophenoxy)acetamido]-1-methylpyrrolidine-2-carboxamide
N-methyl-5-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
7-(2-methoxyethyl)-2-[2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
5-methanesulfonyl-N,2-dimethyl-N-[2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
5-methyl-1-[3-oxo-3-(pyrrolidin-1-yl)propyl]-5-phenylpiperidin-2-one
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
4-methyl-2-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}phenol
6-(furan-3-yl)-2-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
(1S,5R)-3-(naphthalen-2-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(5-acetylthiophen-3-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-methyl-1-(naphthalen-1-ylmethyl)-N-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
1-[2-(5-{8-methylimidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-3-yl)ethyl]pyrrolidin-2-one
2-{1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]pyrrolidin-2-yl}-4-methyl-1H-1,3-benzodiazole
(3R,5S)-5-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrrolidin-3-ol
N-[(3-hydroxypyrrolidin-3-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-(2-methoxyethyl)-5-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}pyrimidine