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6-(benzyloxy)-1-(oxan-4-ylmethyl)-4-[3-(pyridin-2-yl)propanoyl]-1,4-diazepan-2-one
4-({5-[1-(2-phenylethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(2-chlorophenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{1,9-dioxaspiro[5.5]undecan-4-yl}acetamide
N-[(1-phenylpiperidin-4-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(dimethylamino)-3-(4-{[methyl({[2-(trifluoromethyl)phenyl]methyl})amino]methyl}phenoxy)propan-2-ol
2-{[6-oxo-1-(3-phenylpropyl)piperidin-3-yl]formamido}acetamide
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-oxaspiro[4.5]decan-2-one
ethyl 4-{3-[({[4-(trifluoromethyl)phenyl]methyl}amino)methyl]-6H,7H,8H-cyclopenta[g]quinolin-2-yl}piperazine-1-carboxylate
3-[(2,3-dimethylquinoxalin-6-yl)formamido]-3-(4-fluorophenyl)propanoic acid
2-cyclopropyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(3,3,3-trifluoropropyl)piperidine-4-carboxamide
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenyl-1H-1,2,3,4-tetrazole
2-[3-(piperazin-1-ylmethyl)phenyl]-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-methylbut-2-en-1-one
1-[3-({[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-benzyl-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
2-(2-hydroxyethyl)-8-[2-(methylsulfanyl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-5-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methoxy-1-{3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
2-(1H-imidazol-2-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
1-(4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}piperidin-1-yl)ethan-1-one
[(3S,5R)-1-(4-chloro-3-fluorobenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
9-[(4-fluorophenyl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-2-ol
2,6-dimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyrimidine-4-carboxamide
3-{[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-(morpholine-4-carbonyl)pyridin-2-amine
N-{1-[1-(2-hydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
2-ethoxy-5-{2-[(1-hydroxypropan-2-yl)amino]pyrimidin-4-yl}benzoic acid
N-(cyclohexylmethyl)-2-(dimethylamino)-2-(3-methylphenyl)acetamide
2-ethyl-N-[(4-methylphenyl)(thiophen-2-yl)methyl]pyrimidine-5-carboxamide
2-[({5-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
4-ethyl-1-[(3-phenylphenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-butyl-4-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperazin-2-one
8-[1-(3,4-dimethoxyphenyl)propan-2-yl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3-chloro-5-fluorobenzoyl)-2-ethyl-1-(propan-2-yl)piperazine
methyl 3-(2-methoxybenzamido)-5-{[(2-methyl-1,3-thiazol-4-yl)formamido]methyl}benzoate
1-ethyl-N-(6-methylpyridin-3-yl)-6-oxopiperidine-3-carboxamide
4-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]-5-methyl-1-propyl-1H-pyrazole
1-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
1-(propan-2-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
2-{4-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
1-methyl-4-[5-(1-methylpyrrolidin-3-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]piperidine
2-[(dimethylcarbamoyl)amino]-N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]acetamide
N-butyl-N-[(3-methylthiophen-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-[4-(3-methoxypyrrolidin-1-yl)piperidin-1-yl]-6-methyl-2-(piperidin-1-yl)pyrimidine