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2-methoxy-3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrazine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
2-(7-methyl-2-oxo-2H-chromen-4-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
2-[2-(pyridin-2-yl)ethyl]-9-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
(1R,3S)-7-[(3-chloro-2-fluorophenyl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
2-[1-(2-chloro-4-fluorobenzoyl)pyrrolidin-3-yl]benzoic acid
2-(4-methoxy-3-methylphenyl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-(5-carbamoyl-2-methylphenyl)-3-(2,6-dimethylphenoxy)azetidine-1-carboxamide
8-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
7-[(3-methoxyphenyl)methyl]-2-(2-methylpropyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 3-{[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]amino}-1-benzothiophene-2-carboxylate
N-[(3S,4R)-1-[2-(benzenesulfonyl)ethyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
(2S,4R)-4-amino-1-(7-chloro-2-methylquinoline-4-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{2-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]ethyl}pyridine-3-carboxamide
4-(cyclopropylmethyl)-N-(furan-2-ylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
2,7,8-trimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}quinoline-4-carboxamide
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{[2-(2-phenylethynyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-(thiomorpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,4-dithiepan-6-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-5-methylthiophene-2-carboxamide
(3aR,6aR)-2-(3-methoxy-2-methylbenzoyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 3-benzyl-1-{[3-(ethoxycarbonyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
N-cyclopropyl-5-(pyrrolidin-2-yl)-N-(1,3-thiazol-5-ylmethyl)thiophene-2-carboxamide
1-methyl-5-[2-(pyridin-4-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-{[6-(dimethylamino)pyrimidin-4-yl]amino}-2-methylheptan-2-ol
[(3R,4R)-4-[(dimethylamino)methyl]-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
6-fluoro-2-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
(2S)-2-amino-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]cyclohexanecarboxamide
4-[(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]piperidin-4-amine
1-cyclopentyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
3-({4-[3-(4-fluoropiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
N4-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
1-(2-{1-benzyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)pyrrolidin-2-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-6-methoxypyrimidin-4-amine
4-chloro-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-pyrrole-2-carboxamide
1-(1-benzofuran-2-ylmethyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{8-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
5-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[1-(trimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]benzoic acid
N-(2-methoxyethyl)-N,5-dimethyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
5-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1'-{[4-(2-hydroxyethoxy)phenyl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(2-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-2,3-dihydro-1,2-benzothiazol-3-one
N-(3,4-dimethylphenyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-amine
5-[3-(3-methylphenoxy)azetidine-1-carbonyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole
5-(3-benzoylpiperidine-1-carbonyl)-2,3-dimethyl-1H-indole