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N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-propoxyacetyl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(dimethylamino)azepan-1-yl]propan-1-one
2-amino-4-(7-hydroxyquinolin-3-yl)-6-(propan-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methylpiperazin-2-one
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-pyrrol-1-yl)pentan-1-one
N-methyl-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
N-(1-carbamoylcyclopentyl)-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
4-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(methylamino)ethan-1-one
5-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
(1S,9R)-11-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(3S,9aR)-3-(propan-2-yl)-8-(thiophen-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3aS,6aS)-2-[(3-chloro-2,4-difluorophenyl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-2-(pyridin-3-yl)piperidine-1-carboxamide
5-(azepane-1-carbonyl)-1-[2-(dimethylamino)ethyl]piperidin-2-one
2-[(isoquinolin-5-yloxy)methyl]-N-[(3-methoxyphenyl)methyl]-1,3-oxazole-4-carboxamide
(3S)-1-[(1-{[1-(6-methylpyridazin-3-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
3-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
3-{4-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-4-oxobutyl}-3,4-dihydroquinazolin-4-one
8-(furan-3-ylmethyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-amino-6-{2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-(5-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
N-[(3S,4R)-1-(1H-indole-2-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-(2-hydroxyethyl)-2-methoxy-N-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-oxo-1-[2-(3-oxopiperazine-1-carbonyl)phenyl]pyrrolidine-3-carboxylic acid
5-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1-(3-phenylpropyl)-4-{[(trimethylpyrazin-2-yl)methyl]amino}pyrrolidin-2-one
3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-[2-(propylsulfanyl)phenyl]urea
1-[(2,6-difluorophenyl)methyl]-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
(1-{[2-(propylamino)pyrimidin-5-yl]methyl}azepan-2-yl)methanol
3-[2-(4-hydroxy-3-methoxyphenyl)ethyl]-3H,4H-pyrido[3,2-d]pyrimidin-4-one
N-(1-{4-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]phenyl}ethyl)acetamide
2-methoxy-N-({3-methyl-7-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-phenylacetamide
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-N-(1-methyl-1H-pyrazol-3-yl)acetamide
3-[2-(4-fluorophenyl)ethyl]-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperidine
N-methyl-3-(5-methylfuran-2-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-[(2-acetamidoethyl)amino]-N-(quinoxalin-6-yl)pyridine-2-carboxamide
2-benzyl-8-(4-methyl-1H-imidazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-(piperazin-1-yl)ethan-1-one
(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)(phenyl)methanol
5-(4-methoxyphenyl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]furan-2-carboxamide
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}azetidin-3-ol
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
4-{[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1H-pyrazole-3-carboxylic acid
(3S)-N,N-dimethyl-1-(2-phenoxybenzoyl)azepan-3-amine