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N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-[4-methyl-2-({[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}amino)pyrimidin-5-yl]ethan-1-one
6-{4-[(dimethylamino)methyl]phenyl}-3,4-dihydroquinazolin-4-one
3-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-1-(dimethyl-1,2-oxazol-4-yl)urea
1-cyclopropanecarbonyl-N-[(6-methylquinolin-5-yl)methyl]piperidine-4-carboxamide
3-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}piperidin-2-one
3-(hydroxymethyl)-1-(5-methylpyridine-3-carbonyl)piperidin-3-ol
2-[ethyl(methyl)amino]-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
4-(3-chlorophenyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
8-cyclopentyl-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,3-dihydro-1H-inden-2-yl)-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-[3-cyclopropyl-1-(2,3-dimethylphenyl)-1H-1,2,4-triazol-5-yl]-1-oxaspiro[4.4]nonan-2-one
(2R,3R,6R)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]propanoic acid
1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
5-methyl-3-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]-1,2-oxazole
4-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyridine
1-[(4-fluorophenyl)methyl]-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
2-methyl-3-[3-(1-methyl-1H-imidazole-2-carbonyl)phenyl]pyrazine
(4aS,8aR)-6-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-{1-[(9-ethyl-9H-carbazol-3-yl)methyl]piperidin-4-yl}-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-[methyl(quinoxalin-2-ylmethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
ethyl 1-(2-methylbut-3-yn-2-yl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
4-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-3-yl}benzoic acid
2-{5-[1-(2,3-dihydro-1H-indene-5-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
(benzylsulfamoyl)[2-(diethylamino)-2-(furan-2-yl)ethyl]amine
[(5-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-(2-hydroxyethyl)-5-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]thiophene-2-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]pyrazolo[1,5-a]pyridine-3-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propan-1-one
1-[2-(1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)ethyl]pyrrolidin-2-one
5-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-4-phenyl-1H-imidazole
4-[3-(4,5-dimethyl-2-oxo-2,3-dihydro-1,3-oxazol-3-yl)propoxy]benzamide
2-(2-fluorophenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
2-[4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl]pyridine
1-(4-fluoro-3-methoxyphenyl)-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
1-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(4-fluorophenyl)methyl]-4-[(4-methoxypyridin-2-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
4-(4-fluorophenyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
N-(1-methyl-1H-indazol-3-yl)-2-[3-(thiophen-3-yl)-1H-pyrazol-1-yl]acetamide
4-{[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}-N-methylbutanamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(3-phenoxypropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(4-phenylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(2S,4S)-4-amino-1-(4-chloro-2,5-dimethylbenzenesulfonyl)-N-methylpyrrolidine-2-carboxamide
2-(4-{3-[(3-aminopyrrolidin-1-yl)methyl]-7-methylquinolin-2-yl}piperazin-1-yl)ethan-1-ol
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile