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[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
1-{5-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N-(2,2-dimethyloxan-4-yl)-5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
1-[(1-{6-[(1-cyclopropylethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
2-ethyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-({5-[(2-methyl-1-benzothiophen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-cyclohexyl-4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1,4-diazepane
5-methoxy-2-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}pyridin-4-ol
N-propyl-N-(pyridin-3-ylmethyl)isoquinoline-1-carboxamide
1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)-4-(2-methylphenyl)piperazine
3-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
1-{4-[({[1-(dimethylamino)cyclohexyl]methyl}amino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]acetamide
2-[1-(6-methoxypyridin-3-yl)-1H-imidazol-2-yl]-1H-1,3-benzodiazole
(2S)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
[3-({1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
(3R,5S)-5-[4-(4-methoxybutyl)piperazine-1-carbonyl]pyrrolidin-3-amine
1-{[(3R,4R)-4-(hydroxymethyl)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methyl}piperidin-4-ol
4-(cyclopropylmethyl)-1-(4-phenylbutanoyl)-1,4-diazepan-5-one
8-(2-ethoxyacetyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1H-pyrazol-1-yl)propan-2-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-{4-[4-(3-methoxypiperidin-1-yl)piperidin-1-yl]phenyl}-5-phenylpentanamide
4-(1H-imidazol-1-ylmethyl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
(4aS,7aR)-1-(1-benzoxepine-4-carbonyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1H-1,2,3-triazol-4-yl)-2-methoxypyridine
2-{[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzonitrile
1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
2-amino-4-(1H-indol-5-yl)-6-[4-(morpholin-4-yl)phenyl]pyridine-3-carbonitrile
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-ethyl-N-methylpiperidine-3-carboxamide
2-amino-6-(2,2-dimethyloxan-4-yl)-4-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
(2E)-3-(3-fluorophenyl)-N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-phenylpyrrolidin-3-yl]-3-methoxypropanamide
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-2,8-dimethylquinoline
2-{2-[1-(1H-1,2,3-benzotriazol-5-yl)-1H-imidazol-2-yl]-4-chlorophenoxy}acetamide
(4aS,7aR)-1-[(2-fluoro-5-methylphenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[methyl({4-[3-(trifluoromethyl)piperidine-1-carbonyl]phenyl})amino]ethan-1-ol
(1S,5R)-3-(pyrimidin-2-yl)-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-4-(trifluoromethyl)pyrimidin-2-amine
N-{1-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
1-(1,3-benzoxazol-2-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)piperidin-4-amine
[3-(cyclopropylmethyl)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methanol
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(piperidine-1-sulfonyl)pyrrolidin-3-amine
N-(2-hydroxybutyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
(2R)-2-amino-2-phenyl-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]acetamide
3-(3-methoxypropyl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidine-3-carboxylic acid