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[(2-ethylpyrimidin-5-yl)methyl]({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amine
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
2-({1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}oxy)-N-cyclopropyl-4-methoxybenzamide
N-benzyl-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
1-[2-(3-chlorophenyl)ethyl]-4-{[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
4-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-4-phenylbutanamide
methyl 4-{[2-(4-methoxyphenyl)phenyl]carbamoyl}piperazine-1-carboxylate
1-(2-hydroxyethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-1,3-benzodiazole-5-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
N-(furan-3-ylmethyl)-N-methyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
7-(1,3-benzothiazol-2-yl)-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1-butylpiperidin-4-yl)methyl]-3-(pyrrolidin-3-yl)benzamide
2-[(4-chlorophenyl)methyl]-8-(3-ethyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-3-phenylpiperazine
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-(pyrazin-2-ylmethyl)pyrimidin-2-amine
8-methoxy-2-{[4-(thian-4-yl)piperazin-1-yl]methyl}quinoline
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1-benzofuran-2-carboxamide
N-[2-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazol-4-yl)ethyl]acetamide
N-(1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
2-{[7-(2-methoxy-6-methylbenzoyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
2-{4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]morpholin-3-yl}acetic acid
2-cyano-N-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(4-fluorophenyl)butan-1-one
1'-(cyclopropylmethyl)-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
(3S,5S)-1-methyl-5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrrolidin-3-amine
5-benzyl-N-{[(1R,2R)-2-hydroxycyclohexyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
3-ethyl-4-methyl-N-[3-(4-methylbenzamido)phenyl]-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(4-fluorophenyl)ethyl]benzamide
1-(3,4-dimethyl-5-sulfamoylbenzamido)cycloheptane-1-carboxamide
6-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-cyclopropyl-2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2-(2,5-dimethoxyphenyl)-N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
N-{1-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}pyridine-3-carboxamide
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-[4-(oxan-2-ylmethoxy)phenyl]-3-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}urea
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(naphthalen-2-yl)piperazine
ethyl 1-{[3-(methylsulfanyl)phenyl]carbamoyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-methyl-6-[4-(2-phenylethyl)piperidine-1-carbonyl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
6-methoxy-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)pyrimidin-4-amine
N6-cyclopentyl-N5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2-(1,3-thiazol-2-yl)piperidine
2-(methoxymethyl)-4-oxo-N-propyl-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
4-fluoro-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
4-{5-[4-(1H-imidazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
2-{2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylpyridine-3-carboxamide