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1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,3-dihydro-1H-inden-2-yl)acetamide
(2S)-2-(2,3-difluorophenyl)-2-[4-(piperidin-1-yl)butanamido]acetic acid
N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
4-ethyl-1-[(3-methylphenyl)methyl]-1,4-diazepan-5-one
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-(pyridin-3-ylmethyl)cyclopropanamine
8-[(3-chloropyridin-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4,6-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(4-{[2-(dimethyl-1,3-thiazol-5-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
3-(azepane-1-carbonyl)-1-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(4-ethoxyphenyl)methyl]-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
(3aR,5S,6S,7aS)-2-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-octahydro-1H-isoindole-5,6-diol
N-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)methanesulfonamide
2-methoxy-N-[1-(2-phenylethyl)-5-(4-phenylpiperazine-1-carbonyl)-1H-1,3-benzodiazol-7-yl]acetamide
4-(3-fluorophenoxy)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-{2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl}-N-methylmethanesulfonamide
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
{3-propyl-1-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidin-3-yl}methanol
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
N-methyl-2-(3-oxo-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)acetamide
1'-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 2-{8-[(4-methoxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
7-(pyridin-3-yl)-4-(trimethyl-1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
14-(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-(hydroxymethyl)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-ol
ethyl 2-amino-3-cyano-4-(4-hydroxy-2-methoxyphenyl)-5,6,7,8-tetrahydroquinoline-6-carboxylate
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-4-phenylpyrimidin-2-amine
(1S,5R)-6-(cyclobutylmethyl)-3-(quinolin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-cycloheptyl-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}morpholine-2-carboxamide
5-[3-(3-fluoro-4-methoxybenzoyl)piperidine-1-carbonyl]quinoxaline
8-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
6-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-2,3-dimethylquinoxaline
[1-(4-aminopyrimidin-2-yl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol
(1S,5R)-6-benzyl-3-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]propanamide
N'-[3-(2-methoxybenzamido)phenyl]-N-(5-methyl-1,2-oxazol-3-yl)ethanediamide
2-(4-fluorophenoxymethyl)-4-hydroxy-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-5-carboxamide
1-[2-(3-fluoro-4-methoxyphenyl)pyridine-4-carbonyl]-4-methylpiperazine
2-amino-4-(6-ethoxypyridin-3-yl)-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
(1S,5R)-3-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-amino-6-methoxypyrimidin-4-yl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(4-methylpiperazin-1-yl)pyridine-3-carboxamide
7-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]-2-phenoxyethan-1-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-(2,3-dimethylphenyl)-2-[(2-hydroxyethyl)(thiophen-2-ylmethyl)amino]acetamide