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3-[2-(morpholin-4-yl)-2-oxoethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
1-(1-benzylpiperidin-4-yl)-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-ethoxypropan-1-one
[3-(2-methoxyethyl)-1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methanol
4-(methylsulfanyl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]benzamide
N-benzyl-N-methyl-1-{2-[2-(pyridin-2-ylsulfanyl)acetamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-[4-(1H-indol-3-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
N,2-dimethyl-5-phenyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
methyl 4-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-(1-methylazepane-2-carbonyl)-4-phenylpiperidine-4-carbonitrile
2-(dimethylamino)-N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-(4-methylphenyl)acetamide
N-(1,3-benzothiazol-6-yl)-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
ethyl 1-[(5-methylthiophen-2-yl)sulfonyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
5-cyclopropyl-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-oxazole-4-carboxamide
3-{[4-(5-chloro-2-methylphenyl)piperazin-1-yl]methyl}-3-hydroxy-1-methylpiperidin-2-one
2-ethoxy-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}benzamide
ethyl 5-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-(5-tert-butyl-1H-pyrazol-3-yl)-1-(3-methoxypropyl)-1H-imidazole
2-(dimethylamino)-2-(4-fluorophenyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-(trifluoromethyl)pyrimidine
9-(5-methyl-1,3-oxazole-4-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]methylamine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylquinoline-2-carboxamide
[(4-fluorophenyl)methyl](methyl){[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(2-methyl-5-propylpyrimidin-4-yl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]piperidin-4-amine
5-(5-methylpyridine-3-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl 6-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]pyridine-2-carboxylate
2-methoxy-1-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-[(5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}furan-2-yl)methyl]-1H-pyrazole
N-(2-methoxyphenyl)-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-(3-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}pyridin-2-yl)acetamide
9-(5-ethyl-1H-pyrrole-2-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-cyclopentyl-5-[3-(1H-pyrazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-cyclopentanecarbonyl-7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
1-cyclohexanecarbonyl-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
1-{4-[(1-propylcyclopropyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N,N-dimethyl-2-({[1,2,3,4]tetrazolo[1,5-a]pyridin-6-ylformamido}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(3aS,6aS)-5-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole
(3aS,6aS)-2-(4-chloro-2-methoxybenzoyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-phenyl-N-({1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}methyl)benzamide
5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2,4-dimethoxyphenyl)-3-[(3S,4R)-4-(dimethylamino)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propanamide
4-[(4-fluorophenyl)methyl]-1-(furan-3-ylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
[(2S,6S)-4-[(2-chloro-4-fluorophenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol