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5-{2-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}-4,5,6,7-tetrahydro-1H-indazole
(3R,4R)-4-(hydroxymethyl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-3-ol
propan-2-yl 3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carboxylate
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-oxopentanamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
5-methyl-N-({1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)pyrazine-2-carboxamide
2-butoxy-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
4-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1-methylpyrrolidin-2-one
3-(4-fluorophenyl)-4-{[4-(furan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
N-(furan-2-ylmethyl)-6-methyl-N-[2-(morpholin-4-yl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
9-[(3-hydroxy-4-methoxyphenyl)methyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-[(2-propoxyphenyl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(1H-1,2,4-triazol-3-yl)benzamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
3-(3-{[3-(pyridin-3-ylmethyl)piperidin-1-yl]methyl}-1H-indol-1-yl)propanamide
2-benzyl-8-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[4.5]decan-3-one
5-cyclobutanecarbonyl-1'-[(3,4-dimethylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 4-[1-(4,6-dihydroxypyridine-3-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
6-fluoro-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
2-({[3-(4-fluorophenyl)oxolan-3-yl]methyl}amino)-4-methylbenzonitrile
5-(3,4-difluorophenoxymethyl)-N-[2-hydroxy-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
1-ethyl-N-(2-methoxyethyl)-5-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
8-(2,2-dimethylpropyl)-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
N-(2-fluoro-4-methylphenyl)-7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepine-2-carboxamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-(2-oxopyrrolidin-3-yl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-cyclopropyl-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-methyl-3-{[methyl(2-phenylethyl)amino]methyl}-1,2-dihydroquinolin-2-one
N-({3-methyl-7-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
2-({1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl}oxy)pyrimidine
methyl 2-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}piperidine-1-carboxylate
2-[1-(2-phenylethyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl]ethan-1-ol
5-cyclopropyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3,4-oxadiazol-2-amine
[(2S)-1-{2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)pyridine-3-carbonyl}pyrrolidin-2-yl]methanol
3-ethyl-1-[3-(morpholin-4-yl)benzoyl]piperidine-3-carboxylic acid
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]urea
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
N-{2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}acetamide
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
3-cyclopropyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
4-ethyl-N-methyl-1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidine-4-carboxamide
(2R)-N-tert-butyl-N-(thiophen-3-ylmethyl)oxolane-2-carboxamide
6-{[4-(3-cyclohexyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}pyrimidin-4-ol
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-1H-1,3-benzodiazole-5-carboxamide
5-(1-cyclopentyl-5-oxopyrrolidine-3-carbonyl)-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide