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1-(4-{4-[(cyclohex-1-en-1-ylmethyl)amino]piperidin-1-yl}phenyl)-3-methylimidazolidin-2-one
ethyl 1-(benzylcarbamoyl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-3-(pyridin-3-yl)propanamide
2-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-ethyl-4-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)morpholine
N-(4-methylphenyl)-2-({[2-(1H-pyrazol-1-yl)phenyl]methyl}amino)propanamide
3-(2-oxo-2-{4-oxo-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-1'-yl}ethyl)imidazolidine-2,4-dione
ethyl 4-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
(2S)-2-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}propanamide
N-(5-{[(2,3-dihydroxypropyl)(methyl)carbamoyl]amino}-2-methylphenyl)cyclopentanecarboxamide
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
(3R,4R)-4-(hydroxymethyl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-ol
{3-[2-(methylsulfanyl)pyridine-3-carbonyl]-9-propyl-3,9-diazaspiro[5.5]undecan-1-yl}methanol
(4aS,8aS)-2-(quinolin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
2-(2-methyl-1,3-thiazol-4-yl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
4-(2-phenylmethanesulfonylbenzoyl)piperazine-2-carboxylic acid
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
8-chloro-N-[2-(pyrrolidine-1-sulfonyl)ethyl]quinoline-2-carboxamide
1-(3-ethynylbenzoyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
5-ethyl-N4-(1H-indol-6-ylmethyl)pyrimidine-2,4-diamine
1-cyclopentyl-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
6-(3-ethoxyphenyl)-9H-purin-2-amine
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[2-methyl-2-(morpholin-4-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
N,N-dimethyl-5-[6-methyl-4-(morpholine-4-carbonyl)quinolin-2-yl]pyrimidin-2-amine
2-(2-hydroxyethyl)-6-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]piperidin-4-amine
9-hydroxy-2-[(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)methyl]-4H-pyrido[1,2-a]pyrimidin-4-one
6-ethyl-N,1-dimethyl-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(furan-2-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2-methoxyethyl)-1,1-dioxo-N-(thiophen-2-ylmethyl)-1λ6-thiane-4-carboxamide
2-[6-(isoquinolin-5-yl)pyridin-3-yl]acetic acid
(3R,5S)-5-(3-fluorophenoxymethyl)-N-[3-(morpholin-4-yl)propyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-(1H-pyrazol-3-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-N-methylacetamide
N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-benzothiazole-5-carboxamide
1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-[(3-methylphenyl)methyl]piperazine
N-[(3R,4S)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
ethyl 4-{[4-(pyridin-2-ylmethoxy)phenyl]carbamoyl}piperazine-1-carboxylate
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(thiophen-2-yl)acetyl]piperidine-4-carboxamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-(pyrrolidin-3-yl)acetamide
4-[4-phenyl-1-(piperidin-4-ylmethyl)-1H-imidazol-5-yl]-2-(propan-2-yl)pyrimidine
methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})(thiophen-2-ylmethyl)amine
3-[(benzylamino)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one