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1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-[4-(4-fluorophenyl)-2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy]ethan-1-one
ethyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]{[2-(prop-2-en-1-yloxy)phenyl]methyl}amine
4-{[4-(5-butylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
4-[3-(5-fluoro-2-methoxyphenyl)-1-methyl-1H-1,2,4-triazol-5-yl]morpholine
1-(4-benzylpiperidin-1-yl)-3-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}propan-1-one
1-ethyl-2,2-dimethyl-4-(3-methylfuran-2-carbonyl)piperazine
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N,N-dimethylpyrimidin-2-amine
1-(isoquinoline-1-carbonyl)-N-phenylpiperidin-3-amine
N-methyl-2-(morpholin-4-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]-2-(pyridin-3-yl)acetamide
N-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)-N-(oxolan-2-ylmethyl)acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
N-(3-carbamoyl-2-methylphenyl)-4-[(methylsulfanyl)methyl]piperidine-1-carboxamide
1-[({3-[(dimethylsulfamoyl)amino]phenyl}carbamoyl)amino]cyclopentane-1-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]propan-1-one
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-methanesulfonylpyrrolidine
N-[3-({[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]acetamide
1-(3-methoxyphenyl)-4-(5-propylthiophene-3-carbonyl)piperazin-2-one
2-[9-(6-cyanopyridin-2-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
(4S)-1-[(4-chloro-2-fluorophenyl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-(2-fluorophenyl)-3-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methylurea
4-({[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl](methyl)amino}methyl)-1-methylpyrrolidin-2-one
2-(carbamoylamino)-N,3-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}butanamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(trifluoromethyl)benzene-1-sulfonamide
4-(benzyloxy)-1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
methyl 5-(3-{[(2-chlorophenyl)formamido]methyl}piperidin-1-yl)-5-oxopentanoate
5-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-7-methylquinolin-3-yl)methanol
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyridin-2-amine
N'-cycloheptyl-N-[2-(dimethylamino)pentyl]butanediamide
2-{4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
2,2-dimethyl-N-({1-[1-(propan-2-yl)piperidin-4-yl]piperidin-4-yl}methyl)propanamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-(3,5-dichlorophenyl)-4-hydroxy-N-[3-(methylamino)propyl]pyrimidine-5-carboxamide
4-{4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1-methylpiperazin-2-one
(1R,5R)-N,N-dimethyl-6-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-benzyl-5-(2,4-dimethoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
N-ethyl-5-{[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-(2,3-dihydro-1H-inden-1-yl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-(3,4-dimethoxyphenyl)-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidin-3-amine
1-benzyl-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
4-cyclopropanecarbonyl-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-[4-(furan-2-carbonyl)piperazin-1-yl]-3-azaspiro[5.5]undecane
1-(1H-1,3-benzodiazole-5-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-6-methoxypyrimidine
2-(1H-pyrazol-1-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}butanamide