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3-[4-(3-methylphenyl)piperazin-1-yl]-N-(2-oxoazepan-3-yl)propanamide
2-chloro-4-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]phenol
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-3-carboxamide
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
N-benzyl-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)methyl]-4-methyl-1,2-dihydrophthalazin-1-one
8-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(1,1-dioxo-1λ6-thian-4-yl)-2-ethyl-N-methylpyrimidine-5-carboxamide
2-amino-6-(3-hydroxyphenyl)-4-(1H-indol-5-yl)pyridine-3-carbonitrile
5-cyclopropyl-1-[4-(furan-2-yl)butan-2-yl]-4-phenyl-1H-imidazole
N-cyclopropyl-6-[4-(2-methoxyethoxy)phenyl]pyridazin-3-amine
1-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2-dihydroisoquinoline-4-carboxamide
2,4-dimethyl-N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}pyrimidine-5-carboxamide
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(2-methylpyrimidin-4-yl)phenyl]piperidine-1-carboxamide
ethyl 4-{3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]-6H,7H,8H-cyclopenta[g]quinolin-2-yl}piperazine-1-carboxylate
4-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}benzene-1-sulfonamide
9-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-6-oxa-9-azaspiro[4.5]decane
cyclopentyl 4-[(6-hydroxy-1,4-oxazepane-4-carbonyl)amino]benzoate
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide
(2S,4R)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
2-(3-methoxypiperidin-1-yl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
{1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
5-[4-(benzyloxy)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
2-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)-6,8-dimethylquinolin-4-ol
2-methoxy-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
1-(3,5-dimethylphenyl)-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]benzoic acid
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
1,3-dimethyl-N-[3-(3-methylpiperidin-1-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-{2-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-4-[(2-methylphenyl)methyl]piperazin-2-one
5-methyl-5-(4-methylpent-3-en-1-yl)-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-2-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyrrolidine-1-sulfonamide
2-{2-[(1,4-dioxan-2-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-benzyl-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-sulfonamide
1-(2,3-dihydro-1H-inden-4-yl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
6-{3-[(3,5-dimethoxyphenyl)methoxy]phenyl}pyrazine-2-carboxylic acid
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)pyridin-2-amine
5-cyclopropanecarbonyl-1'-(1H-indazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1'-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-{[2-(2,3-difluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}-N-methylbutanamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(4aS,8aR)-1-(2-methylpropyl)-6-[3-(1,2-oxazinan-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
7-(2-hydroxyethyl)-2-(3-methylbut-2-enoyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-4-(4-fluorophenyl)-1-[2-(propylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
methyl (2S)-2-{[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-3-yl]formamido}-2-phenylacetate
N-[2-(4-fluorophenoxy)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-butyl-4-(1-methyl-1H-imidazole-2-carbonyl)-1-(3-phenylphenyl)piperazin-2-one