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4-benzyl-1-methyl-3-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(4-cyanobenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
7-[(3-methoxyphenyl)methyl]-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(2-fluorophenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[(1S)-2-hydroxy-1-phenylethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-[(5-ethylfuran-2-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
9-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3-oxo-3-[2-(trifluoromethyl)morpholin-4-yl]propyl}-1,2-dihydropyridin-2-one
1-[2-methoxy-4-(thiomorpholin-4-ylmethyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-[3-(pyridin-2-yl)azetidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-[3-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
(2S,4S)-4-amino-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-N,N-diethylpyrrolidine-2-carboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(4-methoxyphenoxy)piperidine
1-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(naphthalen-2-yl)ethan-1-one
1-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(diphenylmethyl)acetamide
3-[({1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(3-methylbenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
4-{4-[3-(2-methylphenyl)phenyl]-1H-1,2,3-triazol-1-yl}piperidine
4-hydroxy-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxylic acid
6-(4-fluorophenyl)-2-{2-[(3-methoxypiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
9-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-3-azaspiro[5.5]undecane
(3S,4S)-1-[(4-methanesulfonylphenyl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
8-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
4-{1-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]ethyl}pyrimidine
N'-(2,3-dimethylphenyl)-N-(3-hydroxypropyl)-N-methylpropanediamide
(3R,4S)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-amine
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]pyrrolidine-1-carboxamide
N-(2-phenylethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
5-cyclopentyl-3-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,4-dihydropyridine-3-carboxamide
(3S,7S,8aS)-7-{[(2-chlorophenyl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(1R,9S)-5-amino-3-(5-cyano-1-methyl-1H-pyrrol-3-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-[(4-chlorophenyl)methyl]-8-[2-(methylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamido]-N-phenylpiperidine-1-carboxamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-[3-(4-chlorobenzoyl)piperidine-1-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
1-[(4-fluorophenyl)methyl]-4-(quinolin-2-yl)piperazin-2-one
1-{4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carbonyl}piperidin-4-ol
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2,5-dioxo-6-[4-(pyrrolidin-1-yl)butyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]azocane
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyrrolidin-2-yl]methanol
5-methanesulfonyl-2-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidin-4-amine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
2-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one