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7-cyclohexyl-2-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(3,5-dimethylphenyl)-4-(trimethylpyrimidin-4-yl)piperazin-2-one
N-(2-hydroxyethyl)-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-(1,3-thiazol-2-ylmethyl)acetamide
3-[(dimethylamino)methyl]-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-ol
methyl({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})[(2,4,5-trimethoxyphenyl)methyl]amine
4-methyl-2-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)-1,3-thiazole-5-carboxylic acid
4-({3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}carbonyl)benzene-1-sulfonamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
4-[(5-methylfuran-2-yl)methyl]-3-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}piperazin-2-one
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyrazine-2-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[3-(methylsulfanyl)propyl]amine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(furan-3-ylmethyl)piperidine-3-carboxamide
2-[ethyl({[(3R,4R)-1-(2-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-2,2-dimethylpropan-1-one
N-cyclobutyl-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
(4aR,8aR)-2-cyclobutanecarbonyl-7-(pyrimidin-2-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N,1-dimethyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-hydroxy-N-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)pyrazine-2-carboxamide
(3S,4R)-1-(4-cyclopentylpyrimidin-2-yl)-3-methoxypiperidin-4-amine
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-4-(piperidin-1-yl)butanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-tert-butyl-5-(cyclopentylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
N-tert-butyl-4-{4-[(propan-2-yl)amino]pyrimidin-2-yl}benzene-1-sulfonamide
(2E)-N-cyclopropyl-3-(3-fluorophenyl)-N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}prop-2-enamide
N-methyl-3-(piperidin-3-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
(3S,9aR)-8-(naphthalene-1-sulfonyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aR,7aS)-1-(2-methoxyethyl)-4-(pyrimidin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-phenylethyl)piperidine
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-(2-chlorobenzoyl)-N-(pyridin-3-yl)piperidine-4-carboxamide
2-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-azaspiro[4.4]nonan-3-one
ethyl 4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-amido]piperidine-1-carboxylate
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
3-(4-methoxyphenyl)-1-[4-(3-methylpyridin-4-yl)piperazin-1-yl]prop-2-yn-1-one
3-chloro-2-methyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]benzene-1-sulfonamide
(3S,9aR)-3-ethyl-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
4-[(4-fluorophenyl)methyl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-1-(oxan-4-yl)piperidine-4-carboxamide
1-[3-(dimethylamino)pyrazin-2-yl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-(2,5-dioxoimidazolidin-1-yl)-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
N-[(3R,4R)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide