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5-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}pyrimidin-2-amine
2-{3-[1-(but-2-yn-1-yl)-1H-pyrazol-3-yl]phenyl}-3-chloropyridine
2-amino-4-cyclopropyl-6-(3,4-difluorophenyl)pyridine-3-carbonitrile
4-(4-chlorophenoxy)-4-(piperidine-1-carbonyl)piperidine
3-{3-[(2-fluoro-5-methylphenyl)carbamoyl]propanamido}hexanoic acid
3-({4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-[(4aR,7aS)-4-[2-(methylamino)pyridine-4-carbonyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
4-[(diethylamino)methyl]-5-ethyl-N-[(1-methyl-1H-pyrazol-5-yl)methyl]furan-2-carboxamide
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(5-chloro-2-hydroxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
8-(2,3-dihydro-1H-inden-2-yl)-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methoxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidin-4-amine
2-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]-N-methylethane-1-sulfonamide
(3R,4R)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-[4-(2,1,3-benzothiadiazol-5-ylmethyl)piperazin-1-yl]quinazoline
2-(2,4-difluorophenyl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
ethyl 1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
(3R,4R)-1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
6-[(3,3-diphenylpiperidin-1-yl)methyl]-1-methyl-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
(1S,5R)-3-[(2-chloro-6-fluorophenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-(4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-2-hydroxyacetic acid
[1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
2-[4-(3-cyanophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]acetamide
5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
(4aS,7aR)-4-[(5-ethylpyridin-2-yl)methyl]-6,6-dioxo-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(oxan-2-ylmethyl)piperidin-4-yl}methanol
(1S,4S)-5-(2-cyclopentylacetyl)-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}propanamide
[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl](phenyl)methanol
N-{2-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]ethyl}-3-methylpyridin-4-amine
N-[(2-chlorophenyl)methyl]oxolane-3-carboxamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-ethylpiperidine-1-carboxamide
[4-(2-ethoxypyridine-3-carbonyl)-1,4-oxazepan-6-yl]methanol
1-{1-[1-(3-chloro-5-fluorobenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-[(3-fluorophenyl)methyl]-1,4-diazepane
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N,3-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
6-methoxy-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2,3-dimethylphenyl)-2-{[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}acetamide
9-[2-(dimethylamino)butanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-methyl-6-[2-methyl-5-(1,2-oxazol-5-yl)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(5-methylfuran-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
8-methoxy-N-[(2-methyl-1H-imidazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
4-[(4aR,8aS)-6-[2-(2-fluorophenyl)acetyl]-decahydro-1,6-naphthyridine-1-carbonyl]-1-oxaspiro[4.5]decan-2-one
1-(2-ethoxyethyl)-5-[4-(propan-2-yl)piperazine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(furan-2-carbonyl)-4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[benzyl(methyl)amino]-3-(5-{[(cyclopropylmethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol