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1-[(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
5-cyano-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-(2-chloro-6-methylphenyl)-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
3-benzoyl-N-(3-methyl-1-propyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(2S)-4-methyl-2-(methylamino)pentanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,4-oxazepan-6-ol
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-N,N-diethyl-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
(2S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methylpentanamide
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-(quinolin-6-ylmethyl)piperidin-4-amine
1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
4-{1-[1-(5-ethylthiophene-2-carbonyl)piperidin-4-yl]ethyl}morpholine
N,N-dimethyl-3-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrazin-2-amine
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(oxolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
3-{2-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2-ethoxyphenol
N-[(3R,4R)-1-[(5-cyano-1H-pyrrol-3-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}quinoxaline-5-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(naphthalen-1-ylmethyl)benzamide
ethyl 1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-amino-3-ethyl-N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
[(2S)-1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol
N,1,3-trimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(4S)-3,3,4-trimethyl-1-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperidin-4-ol
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
3-[(4-fluorophenyl)methyl]-5-{1-[4-(4-methoxyphenyl)butan-2-yl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
N-[(3R,4S)-1-(6-aminopyrimidin-4-yl)-4-cyclopropylpyrrolidin-3-yl]propane-1-sulfonamide
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
2-(4-methoxyphenyl)-7-methyl-3-[(4-methyl-1,4-diazepan-1-yl)methyl]quinoline
1-(3-{[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}propyl)piperidin-4-ol
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-7-methyl-1-benzofuran-2-carboxamide
2-[4-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
2-(5-ethyl-1,3-oxazole-4-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
N-(5-chloro-2-methoxyphenyl)-3-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)propanamide
3-benzoyl-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
(3S,4S)-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-4-(naphthalen-2-yl)piperidin-3-ol
4-{1-[6-(3-methylphenyl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
N-[(3R,4S)-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methylpyridin-2-amine
N-[2-(3-chlorophenyl)ethyl]-3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
3-benzyl-5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
1,3-dimethyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-(2-oxopyrrolidin-1-yl)benzamide
4-methanesulfonyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]piperazine-1-carboxamide
6-cyclobutyl-2-[3-({methyl[(6-methylpyridin-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
(2R,3S,6R)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(furan-2-yl)-2-hydroxyethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide