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5-(1-ethylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,8-dimethyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(3S,4R)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-cycloheptyl-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidin-4-amine
3-({[6-(dimethylamino)pyridin-3-yl]methyl}(methyl)amino)-1-phenylpropan-1-ol
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[1-(pyrimidin-4-yl)ethyl]urea
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methoxyphenyl)ethyl]acetamide
ethyl 4-(2-phenoxyethyl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
2,6-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylpyrimidine-4-carboxamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(2-methoxypyridin-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
3-{1-[1-(4-methoxyphenyl)piperidin-4-yl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
4-(piperidin-3-yl)-6-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidine
(1,4-dioxan-2-ylmethyl)({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-(3-methyl-3-phenylbutanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-oxo-1-{2-[4-(propan-2-yloxy)phenyl]ethyl}pyrrolidine-3-carboxylic acid
N-[4-(4-methylpyridin-3-yl)phenyl]acetamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(thiophen-3-yl)propan-1-one
2-(2-chlorophenyl)-N,3-dimethyl-N-(1,2-oxazol-5-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
{4-[(2,4-diethoxy-3-methylphenyl)methyl]morpholin-3-yl}methanol
2-ethyl-9-[(1-propyl-1H-pyrazol-5-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-(4-fluorophenoxymethyl)-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
[(5-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-(2H-1,3-benzodioxol-5-yl)-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
benzyl({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N'-(2-ethoxyphenyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]propanediamide
2,2-dimethylpropyl 2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
3-(4-fluoro-3-methylphenyl)-1-(pyridin-3-ylmethyl)-6-(pyridine-4-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(3R,4R)-4-{4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}oxolan-3-yl]piperidine
1-(2-{[(2-methyl-6-propylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
3-{ethyl[(5-ethylpyridin-2-yl)methyl]amino}-1λ6-thiolane-1,1-dione
N-[2-(1-methylpiperidine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-2-[4-(5-ethylpyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]propan-1-one
2-(2-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
1,3-dimethyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[(diethylamino)methyl]-5-ethyl-N-[(5-methylpyrazin-2-yl)methyl]furan-2-carboxamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
4-methyl-3-({2-[2-(trifluoromethyl)morpholin-4-yl]acetamido}methyl)benzoic acid
1-(3-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
3-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[(3,5-dichloropyridin-4-yl)methyl]-3-[(dimethylamino)methyl]piperidin-3-ol
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
9-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-(1-benzylcyclopropyl)-1-(furan-2-ylmethyl)piperidine-3-carboxamide
N-ethyl-N-[(2-fluorophenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-methyl-4-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine