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(1R,5R)-3-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
5-(3-phenoxyphenoxy)-1-azabicyclo[3.2.1]octane
N-methyl-5-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
1-cyclohexyl-3-(2-methoxyethyl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
6-cyclopentyl-1-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclopentyl-5-cyclopropyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
6-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-(propan-2-yl)pyrimidin-4-amine
4-(azepan-1-yl)-N-[2-(diethylamino)ethyl]pyridine-2-carboxamide
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
2-methyl-9-[1-(2-methylphenyl)piperidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(5-methyl-1H-pyrazol-1-yl)acetamide
5-(piperidin-1-ylmethyl)-2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridine
3-[methyl({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]-1-phenylpropan-1-ol
2-hydroxy-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-3-methylbutanamide
7-(cyclopropylmethyl)-2-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2-hydroxyethyl)-8-[2-(pyridin-2-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy]-1-[4-(pyridin-2-yl)piperazin-1-yl]ethan-1-one
1-[3-(2-ethylphenoxy)azetidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
2-[(2,2-dimethyloxan-4-yl)(methyl)amino]-N,N-bis(prop-2-en-1-yl)acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
1-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-methoxyethan-1-one
(3aS,6aS)-2-(2-methoxyacetyl)-5-[(1-methyl-1H-indol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-cyclopentyl-2-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
5-(2-fluorophenyl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[1'-(6-methylpyridazin-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-methoxy-4-[8-methoxy-3-(1H-pyrazol-1-ylmethyl)quinolin-2-yl]phenol
1-(pyrrolidin-1-yl)-3-{1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl}propan-1-one
2-(2-{[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(1R,2R,6S,7S)-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,4-diazepan-5-one
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
5-methyl-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-indazole
(3aR,6aS)-2-methyl-5-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridine
1-cyclopropyl-3-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-1-(1,3-thiazol-2-ylmethyl)urea
(3S,7S,8aS)-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(6-methoxypyrimidin-4-yl)-N-methylpiperidin-3-amine
7-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-cyclobutanecarbonyl-3-[2-(2-fluorophenyl)ethyl]piperidine
1-propyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1H-pyrazole-5-carboxamide
(2S)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
methyl 6-{[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}pyridine-3-carboxylate
3-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-(furan-2-ylmethyl)propanamide
6-methyl-2-(oxan-4-ylmethyl)-5-[5-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(1-benzoxepine-4-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyridine
5-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
(2-{2-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
3-{1-[3-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl}phenol
N-(3-methoxyphenyl)-4-[3-(1,2-oxazolidin-2-yl)propanamido]benzamide