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N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(2-{[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
N-[2-(1H-pyrazol-1-yl)ethyl]-2-{4-[2-(pyridin-2-yl)acetyl]morpholin-3-yl}acetamide
2-(2,5-dimethylphenoxy)-N-[2-(methylsulfamoyl)ethyl]propanamide
3-butyl-1-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
2-{2-[1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
4-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}piperazine-1-sulfonamide
3-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-2,6-dimethylquinoline
2-{1-[(5-methylfuran-2-yl)methyl]-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-amino-6-(4-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
ethyl 1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-3-carboxylate
1-[5-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
5-({[2-(1H-indol-1-yl)ethyl](methyl)amino}methyl)pyrimidin-2-amine
(3R,4R)-4-{[4-methyl-7-(methylsulfanyl)quinolin-2-yl]amino}piperidin-3-ol
1-methyl-N-[3-(methylamino)propyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
5-[1-(furan-3-carbonyl)piperidin-4-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
(1S,5R)-3-benzoyl-6-(cyclopropanesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-[(3-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)piperidine-4-carboxamide
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-2-carboxylic acid
2-(4-fluorophenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
3-chloro-4-fluoro-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-benzothiophene-2-carboxamide
3-(4-methyl-3-phenylpiperazine-1-carbonyl)-6-(propan-2-yl)-1,2-dihydropyridin-2-one
{7-[5-(morpholine-4-carbonyl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-{[4-(aminomethyl)piperidin-1-yl]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[2-(propylsulfanyl)ethyl]propanamide
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
N-[2-(azepan-1-yl)ethyl]-N-methyl-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
N-({7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
N-[3-(phenylsulfanyl)propyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
(3aR,6aR)-2-(6-chloropyridazin-3-yl)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3S,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
3-(azepane-1-sulfonyl)-5-(2,3-dihydro-1,4-benzodioxin-6-yl)benzoic acid
N2,N2-dimethyl-N4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
4-methoxy-6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyrimidin-2-amine
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
7-(4-fluorophenyl)-2-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(4-benzyl-1H-pyrazol-5-yl)-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[(1R,2S)-2-phenylcyclohexyl]propanamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}propanamide
2-methyl-4-(4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}phenyl)butan-2-ol
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[3-(dimethylamino)propyl]-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
2-(cyclopropylmethyl)-5-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
(2-{2-[1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
(3R,4R)-1-(3-cyclopentylpropyl)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
3-[(3R,4S)-1-(4,6-dimethoxypyrimidin-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol