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1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-ol
[1-(1H-imidazol-1-yl)propan-2-yl]({[1-(morpholin-4-yl)cyclohexyl]methyl})amine
5-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-cyclopentyl-4-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-4-oxobutanamide
6-(4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine-2,4-diamine
N-[(3-fluorophenyl)methyl]-4-hydroxy-4-[(2-methoxyacetamido)methyl]azepane-1-carboxamide
2-(azepan-1-yl)-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]acetamide
2-[1-(2-benzyl-1,3-thiazol-4-yl)-N-methylformamido]-2-(pyridin-3-yl)acetic acid
propan-2-yl 2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carboxylate
N-[(3S)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-yl]acetamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(1H-indol-3-ylmethyl)piperidin-3-ol
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1H-indazole-3-carboxamide
2-(3,4-dichlorophenyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]morpholine
3-cyclopropyl-5-[4-(1H-pyrrol-1-yl)phenyl]-1H-1,2,4-triazole
4-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-4-oxobutane-1-sulfonamide
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
{[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(6-methylpyridin-2-yl)methyl]amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-cyclopropyl-N-ethylacetamide
3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
N-methyl-3-[N-methyl-1-(2-oxo-6-phenyl-1,2-dihydropyridin-3-yl)formamido]propanamide
5-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyrazine-2-carboxylic acid
3-({4-[(6-cyclopropylpyrimidin-4-yl)amino]piperidin-1-yl}methyl)phenol
4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(3,4-dimethoxybenzenesulfonyl)piperidine
N-[2-(dimethylamino)ethyl]-1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-[methyl(2-phenylethyl)amino]-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
methyl (1R,3S,3aR,6aS)-3-(2-fluoro-4-methoxyphenyl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
5,7-dimethyl-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-(2-fluorophenyl)-2-({2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}formamido)acetic acid
(1S,6R)-3-methyl-9-(morpholine-4-sulfonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
(3aS,6aS)-2-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
{1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]quinoxaline
5-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
4-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-3-methoxypropan-1-one
1'-(3-hydroxy-4-methoxybenzoyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-(4-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}phenyl)acetamide
(1R,5R)-6-propyl-3-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-3-[5-(5-methylpyrazine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
1'-(1-tert-butyl-5-oxopyrrolidine-3-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-4-(pyridin-2-yl)pyrimidin-2-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2,6-dimethylquinoline-4-carboxamide
2-[2-(6-chloro-1H-1,3-benzodiazol-2-yl)phenoxy]acetamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-(methylsulfanyl)benzamide
methyl 2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate