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2-(4-fluorophenoxymethyl)-5-[2-(hydroxymethyl)piperidine-1-carbonyl]pyrimidin-4-ol
N-(1H-1,3-benzodiazol-2-yl)-2-{[1-(pyrazin-2-yl)propan-2-yl]amino}acetamide
(3S,4S)-4-(1H-imidazol-2-yl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
5-methoxy-N,1-dimethyl-N-[3-(oxolan-2-yl)propyl]-1H-indole-2-carboxamide
6-(6-hydroxy-1,4-oxazepane-4-carbonyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
5,6-dimethyl-2-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
2-ethoxy-5-[2-({2-[(2R)-pyrrolidin-2-yl]ethyl}amino)pyrimidin-4-yl]benzoic acid
1-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
2-(ethylamino)-N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}pyrimidine-5-carboxamide
propyl 8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
3-(3,4-difluorophenyl)-1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}propan-1-one
(3R,4S)-4-[4-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
(3S,4R)-1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
(3S,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(cyclohexylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
4-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
ethyl 2-(4-{[cyclopropyl(1,3-thiazol-2-ylmethyl)carbamoyl]amino}phenyl)acetate
2-[4-(3,5-difluoropyridine-2-carbonyl)piperazin-1-yl]-1,3-benzothiazole
4-({5-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
methyl[(5-methylfuran-2-yl)methyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
(1R,9aR)-1-({[(2R)-oxolan-2-ylmethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-[(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
6-(2-methoxyphenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyridazin-3-amine
2-[4-(4-chlorophenyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
1-methyl-4-{[5-(oxan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
N-methyl-N-{2-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
4-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-1-oxaspiro[4.5]decan-2-one
6-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
5-chloro-N-(3,4-dihydroxybutyl)naphthalene-1-carboxamide
2-amino-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
(1S,5R)-6-[5-(3-methoxyphenyl)furan-2-carbonyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-[2-methyl-2-(pyrrolidin-1-yl)propyl]-5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazole
(3aS,6aS)-5-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(4-chlorophenyl)ethyl]-N-[(5-ethylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-(3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}phenyl)propanamide
4-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(thian-4-yl)piperidin-3-amine
1-(1-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperidin-4-yl)piperidin-4-ol
2-{[4-(3-methylpyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-{[3-methyl-7-(5-propyl-1,2-oxazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
3-[(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}pyrrolidin-3-yl)methyl]benzamide
9-(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl}-N-(1-phenylethyl)propanamide
2-(4-methoxy-3-methylphenyl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
3-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidine-1-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
10-oxo-N-(4-phenylphenyl)-3,9-diazaspiro[5.6]dodecane-3-carboxamide
2-cyclopropyl-4-methyl-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide