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4-(5-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
4-({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)-1-phenylpyrrolidin-2-one
2-(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}azetidin-3-yl)pyridine
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)(quinolin-4-ylmethyl)amine
(2S,4S)-1-cyclohexyl-N-ethyl-4-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetamido]pyrrolidine-2-carboxamide
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-2-(methylsulfanyl)acetamide
8-(1,3-benzothiazole-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2S,4R)-4-amino-N-methyl-1-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine-2-carboxamide
{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amine
1-(furan-3-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
(3-ethyl-1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-3-yl)methanol
{[4-(butan-2-yloxy)-3-ethoxyphenyl]methyl}(1H-imidazol-2-ylmethyl)amine
2-[1-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-(3-chloro-4-hydroxyphenyl)-1-[3-(2-methylphenoxy)azetidin-1-yl]ethan-1-one
2-(4-cyclohexylpiperazin-1-yl)-2-(3,4-dimethoxyphenyl)acetic acid
2-(morpholin-4-yl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
N-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-4-(furan-3-carbonyl)-1,4-diazepane-1-carboxamide
N-[(5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
2-methyl-3-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-indole-5-carbonitrile
ethyl 1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
(2S)-2-{[(6-cyanopyridin-3-yl)carbamoyl]amino}-3-methylbutanamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(5-ethyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(piperidin-1-yl)-2-(4-{[2-(trifluoromethyl)morpholin-4-yl]methyl}phenoxy)ethan-1-one
5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyridine-2-carbonitrile
(1S,2R)-2-{[(5-fluoro-3-methyl-1H-indol-2-yl)methyl](methyl)amino}cyclohexan-1-ol
N-[4-(3-fluorophenyl)phenyl]-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
methyl[(4-methyl-1H-imidazol-5-yl)methyl][(3-phenyl-1H-pyrazol-4-yl)methyl]amine
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
2-methyl-6-(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-4-yl)pyrimidin-4-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(3-fluorophenyl)methyl]-N-methylpyrimidin-2-amine
N-methyl-4-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-3,4-dihydroquinazoline-2-carboxamide
(4aS,7aR)-1-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-4-cyclopropyl-1-(2-ethoxyethyl)pyrrolidin-3-yl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
4-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(1,2-oxazol-5-yl)phenol
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(dimethyl-1,2-oxazol-4-yl)propanamide
{4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenyl}methanol
1-tert-butyl-5-oxo-N-{2-[4-(trifluoromethyl)phenyl]ethyl}pyrrolidine-3-carboxamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
[(3R,4S)-1-[(4-chloro-2-fluorophenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-methylpropyl)acetamide
(2S)-2-amino-3-(4-hydroxyphenyl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]propanamide
(2S,4R)-4-amino-1-[(6-chloro-2H-chromen-3-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(4-{[methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})amino]methyl}oxan-4-yl)methanol
4-[(cyclopropylmethyl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
2-methyl-4-(4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}phenyl)butan-2-ol