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N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
6-(2-chlorophenyl)-2-[4-(piperidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2-{2-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2-dihydroisoquinolin-1-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
3-methoxy-2-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)phenol
1-[3-(dimethylamino)phenyl]-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methylurea
4-(4-chlorophenyl)-1-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]butan-1-one
methyl 4-[5-methyl-4-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-1,3-oxazol-2-yl]benzoate
4-({5-[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
2-{[4-(cyclopentyloxy)phenyl]methyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(thiophen-3-yl)acetamide
1-[7-(3-fluorobenzoyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidine
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyridin-2-amine
(1R,5S,6R,7S)-3-methyl-6-(3-oxo-4-phenylpiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-phenyl-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-amine
1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-{4-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N,5,6-tetramethylpyrimidin-2-amine
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
4-({2-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(2,5-difluorophenyl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-(1,3-dihydroxypropan-2-yl)-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
2-({[(3S,5S)-1-benzyl-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-yl]amino}methyl)phenol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperidin-3-ol
(4aS,7aR)-1-(2-hydroxypyridine-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{5-[(1-propyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)[(1-methyl-1H-imidazol-5-yl)methyl]amine
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
2-[5-cyclopropyl-4-(4-phenylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
4-[(3-chloro-4,5-dimethoxyphenyl)methyl]-1-phenylpiperazin-2-one
5-chloro-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pyridine-2-carboxamide
2-{[(9H-purin-6-yl)amino]methyl}adamantan-2-ol
2-cyclopentyl-8-(5-methoxypyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-N-ethyl-4-[3-(4-hydroxyphenyl)propanamido]-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
N-(adamantan-1-yl)-3-oxo-3-[2-(pyridin-2-yl)pyrrolidin-1-yl]propanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
2-(4-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
6-(difluoromethyl)-2-{2-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
N-cyclopropyl-N-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
N-methyl-4-(4-methylphenyl)-N-(1H-pyrazol-3-ylmethyl)-5-(pyridin-3-yl)pyrimidin-2-amine
1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
(2R)-2-amino-4-methyl-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pentan-1-one
7-[(3,4-difluorophenyl)methyl]-2-(1,2,3-thiadiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1,4-oxazepane
2-methoxy-N-[1-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N,N-diethyl-1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide