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1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
N-[(4-phenyloxan-4-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
7-(2-methoxyethyl)-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-(cyclopropylmethyl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2S)-2-amino-1-[4-(4-methoxyphenoxy)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
({1-[(2-fluorophenyl)methyl]-2-methyl-1H-indol-3-yl}methyl)({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl})amine
5-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-(2,4-dimethylphenyl)-3-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}propanamide
1-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-3-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-[(1s,4s)-4-aminocyclohexyl]-N-[(4-sulfamoylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[4-(hydroxymethyl)benzoyl]-decahydro-1,6-naphthyridin-2-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(butan-2-yl)acetamide
3-[4-(difluoromethoxy)-2-methylphenyl]-1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)urea
3-(cyclopropylmethyl)-1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidine-3-carboxylic acid
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(1H-pyrazol-3-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(1-{1-[(2R)-2-amino-3-methylbutanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
N,N-dimethyl-2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethane-1-sulfonamide
2-{4-[4-(pyridin-2-yl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-ol
N-(4-fluoro-2-methylphenyl)-3-[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]propanamide
1-(cyclohexylmethyl)-6-oxo-N-propyl-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-{2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}azepan-2-one
(2S)-1-acetyl-N-[(3-chloro-1-benzothiophen-2-yl)methyl]pyrrolidine-2-carboxamide
4-[3-(pyridin-3-yl)propyl]-2-(trifluoromethyl)morpholine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
(3aS,7aR)-5-methyl-2-(5-propylthiophene-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]benzamide
5-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(1-{6-[benzyl(methyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
N-[2-(2-fluorophenoxy)ethyl]-2,4-dimethylpyrimidine-5-carboxamide
N5-[4-(ethylsulfanyl)phenyl]-N2-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2,5-dicarboxamide
1-cycloheptyl-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(4-propylpyrimidine-5-carbonyl)thiomorpholine
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-imidazol-2-yl]-2-(pyrrolidin-1-yl)pyrimidine
3-[3-(2-ethylphenoxy)azetidin-1-yl]-6-methylpyridazine
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-4,6-dimethylpyrimidin-2-amine
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
[(2R)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]methanol
1-benzyl-5-(pyridin-3-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aS,6aS)-N-(3-benzylphenyl)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carboxamide
2-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(2-methoxyquinolin-3-yl)methyl]piperidin-3-ol
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1,3-benzothiazole
(1S,5R)-6-(cyclopropylmethyl)-N-(furan-2-ylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)thiophene-2-carboxamide
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-(2-methoxybenzoyl)-4-[(3-methylphenyl)methyl]-1,4-diazepan-5-one