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1-(3-chloro-4-fluorobenzoyl)-3-(3-methoxypropyl)piperidine
1-[cyclohexyl(methyl)amino]-3-[3-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-{[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}-N-methylpropanamide
N-(2-hydroxyethyl)-5-(3-methoxyphenoxymethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-ethyl-3-[(1E)-pent-1-en-1-yl]benzamide
3-{2-[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
1-(2,2-dimethylpropyl)-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
3-cyclopropyl-5-(2-ethylhexyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)quinoline
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-indazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
4-[(2-fluorophenyl)methyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)-3-oxopiperazine-1-carboxamide
N,2-dimethyl-4-phenyl-N-(thiophen-3-ylmethyl)pyridine-3-carboxamide
2-(2-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
4-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydroquinolin-2-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(propan-2-yl)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidine-2-carboxamide
5-({cyclopropyl[(3-methylthiophen-2-yl)methyl]carbamoyl}amino)-2-methoxy-N-methylbenzamide
3-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]phenol
3-(2-methoxyphenyl)-1-methyl-3-{2-oxo-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
2-({2-[4-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}amino)-6-methyl-3,4-dihydropyrimidin-4-one
3-({1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}methyl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2S,4S)-2-{[(dimethylsulfamoyl)amino]methyl}-4-fluoropyrrolidin-1-yl]-3-(2-fluorophenyl)propan-1-one
1-(2-methoxyphenyl)-2,2-dimethyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazine
N-[2-(4-methoxyphenyl)phenyl]-1-propanoylpyrrolidine-2-carboxamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methoxypiperidine
2-ethyl-9-(1-methyl-1H-pyrrole-2-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
7-(1,3-benzothiazol-2-yl)-4-[(3,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(carbamoylmethyl)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidine-3-carboxamide
ethyl 2-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]acetate
2-{6-[(2-hydroxyethyl)amino]pyridazin-3-yl}-N,N-bis(propan-2-yl)benzamide
2-{[(2-amino-5-methylpyrimidin-4-yl)(methyl)amino]methyl}-2-ethylbutan-1-ol
2-{8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
3-(4-methanesulfonylphenyl)-4-methoxybenzamide
8-fluoro-2-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[(4-fluorophenyl)(hydroxy)methyl]-1H-1,2,4-triazol-3-yl]acetamide
3-(2-methylphenyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
(3S,9aR)-3-[(2S)-butan-2-yl]-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}thian-4-amine
5-ethyl-2-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}pyridine
methyl 2-{[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]amino}benzoate
5-(azepane-1-carbonyl)-N-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-methyl-5-(2,3,5,6-tetramethylbenzenesulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3S,4S)-1-[(1-methylpiperidin-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-methyl-1H-pyrrole-2-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-(thiomorpholin-4-yl)acetic acid
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-{[4-(4-methoxy-2,5-dimethylphenyl)-1H-1,2,3-triazol-1-yl]methyl}-4,6-dimethylpyrimidine
1-benzyl-5-(furan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
3-[4-(dimethylamino)phenyl]-1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
5-fluoro-4-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]quinazoline