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N-[(3S,4R)-1-(4-oxo-4-phenylbutanoyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
5-hydroxy-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrazine-2-carboxamide
6-(benzyloxy)-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
2-(4-{[4-(benzyloxy)-2-methoxyphenyl]methyl}morpholin-2-yl)ethan-1-ol
3-hydroxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
6-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
1-methyl-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2-phenylpiperazine
3-(1H-1,3-benzodiazol-2-yl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}propanamide
2-{2-[4-fluoro-3-(trifluoromethyl)phenyl]phenyl}-5-methyl-1,3,4-oxadiazole
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)(1H-pyrazol-3-ylmethyl)amine
4-(5-methylpyridin-2-yl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-ol
1-[4-(4-hydroxyphenyl)butan-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[(3R,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(2-hydroxyethyl)-8-[2-(pyridin-2-ylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-({3-[1-(dimethylamino)ethyl]phenyl}methyl)-4-phenylpiperidine-4-carbonitrile
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-(2-methoxyethyl)-1-[(2-phenylethyl)carbamoyl]piperidine-3-carboxylic acid
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-cyclopropyl-6-oxo-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,6-dihydropyrimidine-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{6-[(dimethylamino)methyl]pyrazin-2-yl}piperidin-3-ol
3-[1-(4-acetamidobenzenesulfonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
N-methyl-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
N-(diethyl-1,2-oxazol-5-yl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
5-(2,6-difluorophenoxymethyl)-N-(1-hydroxypropan-2-yl)-1,2-oxazole-3-carboxamide
6-(4-{bicyclo[2.2.1]hept-5-en-2-ylmethyl}piperazin-1-yl)pyridine-3-carboxamide
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-6-hydroxy-1,4-oxazepane-4-carboxamide
2-(2,3-difluoro-4-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-propyl-2-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
4-chloro-N-[2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)ethyl]benzene-1-sulfonamide
2-[5-(3-phenyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-(2,6-dimethylphenyl)-3-[2-(dimethylsulfamoyl)ethyl]urea
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[3-(furan-2-yl)propyl]-1-[4-(3-methylpiperidine-1-carbonyl)phenyl]urea
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(furan-2-carbonyl)piperidine-4-carboxylic acid
1-[3-(methylsulfanyl)propyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(ethoxymethyl)-N-(3-phenylphenyl)pyrrolidine-1-carboxamide
1-{[({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]methyl}cyclohexan-1-ol
11-[2-(2-methoxyphenyl)pyrimidin-5-yl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(2-methylphenyl)methyl]piperazine
4,6-dimethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[2-(dimethylamino)ethyl]-5-(quinoline-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(3-methylthiophen-2-yl)sulfonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]phenyl}-5-methyl-1,3,4-oxadiazole
2-chloro-N-[2-(5-methyl-1,3-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
5-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one