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2-methyl-3-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}quinoxaline
2-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-2,3-dihydro-1H-isoindole
N,N-dimethyl-3-({3-oxo-2-azaspiro[4.4]nonan-2-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
1-[(2,6-difluorophenyl)methyl]-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
6-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]pyridine-3-carbonitrile
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 5-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-methyl-N-(1-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carbonyl}pyrrolidin-3-yl)acetamide
1-[1'-(3,4-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
5-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)quinoxaline
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(3-methylbut-2-en-1-yl)piperidine-4-carboxamide
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-butyl-1,3-dimethyl-2,6-dioxo-N-(3-phenylprop-2-yn-1-yl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
3-{[(2-aminopyrimidin-5-yl)methyl](methyl)sulfamoyl}-N-(butan-2-yl)benzamide
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine
N-[4-(furan-2-yl)butan-2-yl]-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
3-hexyl-8-(3-hydroxybenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S)-3-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)azepan-2-one
3-(methanesulfonylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
6-[1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyrimidin-4-ol
(1S,5R)-6-(2,4-difluorobenzoyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[5-(2-butoxyacetamido)-2-methoxyphenyl]furan-2-carboxamide
2-methyl-4-[5-({[(2-methylphenyl)methyl](prop-2-en-1-yl)amino}methyl)thiophen-2-yl]but-3-yn-2-ol
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
2-(2-methoxyethyl)-8-(9H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(3-methylpiperazine-1-carbonyl)-N-[2-(pyridin-3-yl)ethyl]benzene-1-sulfonamide
2-(dimethylamino)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(2-methylphenyl)ethan-1-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
(3R,4R)-4-amino-1-(8-chloroquinolin-2-yl)piperidin-3-ol
4-(9H-fluoren-2-yl)-1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazole
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyridine-3-carboxamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,2-oxazol-5-ylmethyl)propanamide
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(4-{[2-(2,4-difluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenyl)acetamide
N-{2,2,2-trifluoro-1-[1-(3-fluoropropyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}pyridine-4-carboxamide
2-[4-(1-benzofuran-2-ylmethyl)morpholin-3-yl]acetic acid
5-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 2-(1-{1-[(2-methoxyphenyl)methyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
1-methyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(1H-imidazol-1-ylmethyl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-ol
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
3-ethyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-1H-pyrazole-4-carboxamide
4-(3-carboxybenzenesulfonyl)piperazine-2-carboxylic acid