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3-chloro-4-methoxy-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
N3-cyclooctyl-N5-[1-(4-fluorophenyl)ethyl]-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
1-(2-methoxyphenyl)-3-{1-[1-(3-methoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
ethyl 4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine-1-carboxylate
N-butyl-N,5-dimethyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(3-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-[(4-fluorophenyl)methyl]-2-[(2-methoxypyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-(4-methylphenoxymethyl)-3-(2-phenylethyl)-1H-1,2,4-triazole
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-3-[(dimethylamino)methyl]piperidin-3-ol
4-[5-fluoro-2-(4-methanesulfonylphenyl)pyrimidin-4-yl]morpholine
N-[(3R,5S)-5-[4-(pyridin-4-yl)piperazine-1-carbonyl]pyrrolidin-3-yl]benzamide
(4aR,7aS)-1-methyl-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-N-ethyl-1-[(ethylcarbamoyl)methyl]-4-(furan-3-amido)pyrrolidine-2-carboxamide
1-(1-benzylpiperidin-4-yl)-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
(3R,4R)-4-amino-1-[(3-chloro-4,5-diethoxyphenyl)methyl]piperidin-3-ol
2-methyl-2-[4-(oxan-2-ylmethyl)phenyl]propanamide
1-{4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(1H-indol-3-yl)acetamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidine
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-(pyridazine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-benzyl-5-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}pyrimidin-2-amine
{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}(pyridin-2-yl)methanol
1-(1-methanesulfonylpyrrolidine-2-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-(cyclohexylmethyl)-N-[(1-ethylpiperidin-3-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[3-(pyridin-2-yl)propyl]pyrimidin-2-amine
7-phenyl-2-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N3-(2,2-dimethyloxan-4-yl)-1-[(2-methoxyphenyl)methyl]-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-hydroxyethyl)-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
(4aS,8aR)-6-(2,3-dihydro-1H-indene-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(2R,6R)-4-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(4aR,7aS)-4-(5-ethyl-1,3-oxazole-4-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-[(4-chlorophenyl)methyl]-8-(pyridine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
3-amino-3-(3,4-dimethoxyphenyl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-(methoxymethyl)-5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}pyrimidine
(3S,4R)-3-ethyl-4-methyl-1-(3-methylpyrazin-2-yl)piperidin-4-ol
(1H-1,3-benzodiazol-2-ylmethyl)[(1-ethylpyrrolidin-2-yl)methyl]{[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoxaline
2-[1-(pyrimidin-4-yl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
3-ethyl-6-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
N-methyl-5-oxo-1-(pyridin-3-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxamide
2-[4-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)phenyl]-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
4-(2-{2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)phenol
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
N-[1-(2-methanesulfonylethyl)piperidin-4-yl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(2-methoxyethyl)-1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide