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(2S,4R)-4-amino-N-methyl-1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}pyrrolidine-2-carboxamide
5-(1-benzothiophen-3-yl)-1H-1,2,4-triazole
{5-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]furan-2-yl}methanol
(3R,4R)-3-cyclopropyl-4-methyl-1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
1-[3-(4-{[2-(5-methylfuran-2-yl)ethyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
2,2-difluoro-N-[(1-propyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]-2H-1,3-benzodioxole-4-carboxamide
(2S,4S,5R)-4-[(2-carboxyethyl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
1,3-dimethyl-8-(5-methylpyrimidin-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-{[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]methyl}-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
6-{4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazin-1-yl}-9H-purine
3-[1-(2-phenoxypropanoyl)piperidin-4-yl]-N-phenylpropanamide
2-[4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)piperidin-1-yl]pyridine-3-carbonitrile
1-(2-phenoxyethyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2,2-dimethyloxane-4-carboxamide
N3-cycloheptyl-1-cyclopropyl-4-oxo-N5-(2-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(1-methyl-1H-pyrazol-3-yl)-2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
(1S,5R)-3-(3-chloropyridin-2-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-butyl-3-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-[1-({1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-amine
2,6-dimethyl-4-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)phenyl acetate
1-[2-(dimethylamino)acetyl]-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2,3-dihydro-1H-inden-4-yl)-3-ethylurea
4-[2-(3-methoxypropyl)piperidine-1-carbonyl]pyridin-2-amine
2-[4-(difluoromethoxy)benzenesulfonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-methyl-1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-1,4-diazepan-5-one
1-cyclohexanecarbonyl-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
3-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-6-methoxy-2,3-dihydro-1H-indol-2-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
8-(cyclopropylmethyl)-N-(3,4-difluorophenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-(1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-2-yl)-6-methyl-1H-1,3-benzodiazole
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,3-dimethoxybenzamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
2-(2-methylphenyl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-[2-(1-methylpyrrolidin-2-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carboxylic acid
7-({2-[3-(dimethylamino)propoxy]phenyl}methyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-({[(1R,2R)-2-(benzyloxy)cyclopentyl]carbamoyl}amino)-N,N-dimethylbenzamide
1-(3,5-dimethylphenyl)-4-[4-(methylsulfanyl)benzoyl]piperazin-2-one
N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-(diphenylmethyl)-5-(thiolan-3-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-{4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}-1H-1,2,4-triazole
(5S,9aS,9bS)-5-(5-cyclohexylthiophen-2-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[2-(1,2,4-oxadiazol-3-yl)ethyl]amine
2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
3-(hydroxymethyl)-N-{4-[2-(pyridin-2-yl)ethoxy]phenyl}piperidine-1-carboxamide
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-3-(pyridin-2-yl)propan-1-one
(2R)-2-amino-2-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)acetamide
5-(1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
2-{[5-(1-methylpiperidin-3-yl)-4-phenyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid