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N-[(4-chlorophenyl)methyl]-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(4aS,7aR)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(2-methoxyethyl)-1-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
{4-[2-(dimethylamino)-6-(trifluoromethyl)pyrimidin-4-yl]phenyl}methanol
5-(4-fluorophenyl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(1H-indol-2-yl)phenyl]-1-(oxane-4-carbonyl)piperidine-4-carboxamide
6-ethyl-2-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]quinoline-4-carboxamide
4-(4-methylphenyl)-5-(pyrimidin-5-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrimidin-2-amine
N-[(3S,4R)-4-methoxyoxolan-3-yl]-N'-[2-(methylsulfanyl)phenyl]butanediamide
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methoxyethan-1-one
4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(pyridin-4-yl)ethyl]pyrimidine-5-carboxamide
2-cyclopentyl-9-[(2-fluoro-4-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-1-(1-ethylpiperidin-4-yl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[2-(1H-imidazol-1-yl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-(3-methoxybenzoyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
N-(2-fluoro-4-methylphenyl)-2-{[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]formamido}acetamide
N-methyl-2-(oxan-2-ylmethoxy)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-3-(1H-imidazol-2-yl)piperidine
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
1-(2-methylphenyl)-4-(4-propoxybenzoyl)piperazin-2-one
4-{1-[2-(cyclohex-1-en-1-yl)ethyl]-1H-imidazol-2-yl}-1-methylpiperidine
1-(diethylamino)-3-[2-methoxy-4-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
[(4-ethyl-5-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-5-(methoxymethyl)thiophene-2-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(4-fluorophenyl)butan-1-one
methyl(oxolan-2-ylmethyl)[2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethyl]amine
4-[(2S)-2-hydroxy-3-phenylpropanoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)pyrrolidin-3-yl]-2-(pyridin-4-yl)pyridine
1-(3-chloro-5-fluorobenzoyl)-3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine
2-[2-(1H-imidazol-1-yl)ethyl]-1-(2-phenylbenzoyl)piperidine
4-[3-(oxolan-3-yl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]benzonitrile
2-(4-ethylpiperazin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
2-methyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1-benzofuran-5-carboxamide
5-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyrazin-2-ol
N-(2,3-dihydroxypropyl)-7-fluoro-N,3-dimethyl-1H-indole-2-carboxamide
1-(4-methoxybenzoyl)-4-[4-(pyrrolidin-1-yl)benzoyl]piperazine
3-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
N3-cyclooctyl-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(1,4-dioxan-2-ylmethyl)-2-fluoro-6-methoxybenzamide
4-[(2S)-5-oxopyrrolidine-2-carbonyl]-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,2-oxazole-3-carboxamide
1-(2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}pyrimidin-4-yl)piperidin-4-ol
3-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidine-1-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
(3R,4R)-4-(hydroxymethyl)-1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]piperidin-3-ol
(3S,4R)-4-(hydroxymethyl)-1-(6-methoxy-1-methyl-1H-indole-2-carbonyl)piperidin-3-ol
2-(2-hydroxyethyl)-N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)pyrrolidine-1-carboxamide
3-methyl-1-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-propylurea
2-[2-(3-methoxyphenyl)ethyl]-4-{4-[2-(1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione