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3-methyl-1-(2-methylpropyl)-4-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}piperazin-2-one
7-(cyclopropylmethyl)-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[(4-methoxyphenyl)methyl]-4-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[4-(furan-2-yl)butan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-[2-(4-chlorophenyl)ethyl]-5-methyl-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
3-ethyl-N-{2-[methyl(phenyl)carbamoyl]phenyl}-1,2-oxazole-5-carboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-3-carboxylate
2-[(4-methyl-1,4-diazepan-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N,3,6-trimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1-benzofuran-2-carboxamide
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-(1,4-dithiepan-6-yl)piperidine
2-(5-methyl-1-benzothiophen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-cyclooctyl-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-(2,3-dihydro-1H-inden-2-yl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-[2-(benzenesulfonyl)ethyl]-1-[(3,5-dimethylphenyl)methyl]-1,4-diazepan-5-one
4-[5-(1-propylpyrrolidin-2-yl)thiophene-2-carbonyl]morpholine
2-ethyl-5-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-(2-ethoxyphenyl)-N-(1-methyl-1H-pyrazol-4-yl)piperazine-1-carboxamide
5-methyl-1-[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1H-1,2,3,4-tetrazole
5-[1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-imidazol-2-yl]-3-phenyl-1,2,4-oxadiazole
2-(dimethylamino)-8-(3-ethoxyphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)-N-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-pyrazol-5-yl)acetamide
N-methyl-3-{[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
3-({1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-cyclobutanecarbonyl-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-{[(2,3-difluoro-6-methoxyphenyl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
(3aR,6aR)-2-(cyclopentylcarbamoyl)-5-(pyrazin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
(3S,4S)-1-(6-tert-butyl-2-oxo-2,3-dihydropyrimidine-4-carbonyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
4-(dimethyl-1,2-oxazol-4-yl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
7-fluoro-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[6-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridin-3-yl]ethan-1-one
methyl 1-[(3R,5S)-5-[(2-phenylethyl)carbamoyl]-1-(1-propylpiperidin-4-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3,5,7-trimethyl-2-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-1H-indole
1-{5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}propanoic acid
4-(cyclopropylmethyl)-1-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-[4-(3-hydroxy-3-methylbutyl)benzoyl]-N,N-dimethylpiperazine-1-carboxamide
{1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
5-[1-(2-methyl-1,6-naphthyridine-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
6-butyl-2-[3-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2,3-dimethyl-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]quinoxaline-6-carboxamide
2-(3-fluorophenyl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
5-(2-methylpropyl)-1'-(trimethylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3aS,6aS)-2-[(2-chloro-4-fluorophenyl)methyl]-5-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
2-acetyl-8-(5-carboxy-3-chloropyridin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[2-(1H-imidazol-4-yl)ethyl]-8-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
(3R,4R)-N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethylpyrrolidine-3-carboxamide