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1-(morpholin-4-yl)-3-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-yl}propan-1-one
(2S,4S)-4-amino-N-ethyl-1-(3-phenoxybenzoyl)pyrrolidine-2-carboxamide
4-methoxy-2-[4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]pyrimidine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(pyrimidin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-(methoxymethyl)-5-methyl-N-[4-(5-methylfuran-3-amido)phenyl]-1,2-oxazole-3-carboxamide
2-[4-(hydroxymethyl)phenyl]-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]ethan-1-one
4-hydroxy-N,2-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrimidine-5-carboxamide
7-[(3-methoxyphenyl)methyl]-2-(3-methylbutyl)-2,7-diazaspiro[4.5]decan-6-one
2-({4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-(2-fluoro-5-methylphenyl)-N'-[2-(2-methoxyphenyl)ethyl]butanediamide
2-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]phenol
2,3-dimethyl-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(6-methoxynaphthalen-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]morpholine
(1S,5S)-3-[(2-chloro-6-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-(2-methylprop-1-en-1-yl)-1,2,4-oxadiazole
N-(cyclohexylmethyl)-N-ethyl-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
3-({4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
4-({5-[2-(thiophen-2-yl)-1,3-thiazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
ethyl 1-(3-fluorobenzenesulfonyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-ol
N-(2,3-dihydro-1H-inden-2-yl)-5-methoxy-4-oxo-N-propyl-1,4-dihydropyridine-2-carboxamide
5-cyclobutanecarbonyl-1'-[3-(1H-pyrazol-1-yl)propyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidine-3-carboxylate
ethyl 1-[(3-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
(3S,4R)-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
6-methyl-2-(3-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
6,8-dimethyl-2-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)methyl]quinolin-4-ol
2-hydroxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyridine-3-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}benzamide
7-(oxan-4-yl)-2-[2-(2H-1,2,3-triazol-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
(3R,4R)-1-[(2-methoxyquinolin-3-yl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
6-{1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(piperidin-4-yl)piperidine
8-(4-fluorobenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-cyclopentyl-9-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(dimethylamino)ethyl]-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
methyl 4-[5-(4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]butanoate
(3E)-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-3-en-1-one
(2,4,6-trimethyl-3-{[(5-methylhexan-2-yl)amino]methyl}phenyl)methanol
2,3,4-trimethoxy-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
methyl[(5-methyl-1,3-diphenyl-1H-pyrazol-4-yl)methyl][(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
N,N-dimethyl-7-(5-methylpyridine-3-carbonyl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[2-(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
1-(3-oxo-3-{spiro[azepane-4,2'-chromene]-1-yl}propyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-(morpholin-4-yl)propyl]-3-(3-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)urea
1-cyclopentanecarbonyl-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
2-ethyl-6-{1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
8-(6-methyl-2-propylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid