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[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-4-(trifluoromethyl)benzamide
N-(2-methoxyethyl)-4-[2-(methylsulfanyl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1-methyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-2H-1,3-benzodioxole-5-carboxamide
{3-propyl-1-[4-(trifluoromethyl)benzoyl]piperidin-3-yl}methanol
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)propanamide
4-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4H-1,2,4-triazole
9-[(1-methylpiperidin-3-yl)methoxy]-4-[(6-methylpyridin-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})[2-(pyridin-2-yl)ethyl]amine
3-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)propane-1,2-diol
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)pyrimidin-4-yl]pyrrolidin-3-ol
1-(2-{[2-(1H-indol-3-yl)ethyl]amino}pyrimidin-4-yl)piperidin-3-ol
1-cyclopropyl-4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]pyrrolidin-2-one
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
5-{3-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]propyl}-4-methyl-1,3-thiazole
1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
1-ethyl-4-[4-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}piperidin-1-yl)benzoyl]piperazine
4-cyclopentyl-11-[(2-methylpropyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[(1R,3S,3aS,6aR)-5-ethyl-3-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-1-(hydroxymethyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
N-(3-methoxyphenyl)-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
3-[2-(morpholin-4-yl)-2-oxoethyl]-4-(naphthalen-1-ylmethyl)piperazin-2-one
1-{[(3R,4R)-1-(3-fluoropyridin-4-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
5-acetamido-1-(2-methoxyethyl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[4-(hydroxymethyl)phenyl]methyl}acetamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2,6-dihydroxybenzamide
1-{4-methyl-2-[(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)amino]pyrimidin-5-yl}ethan-1-one
5-(methoxymethyl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
4-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-1-(pyridin-2-yl)ethyl}morpholine
8-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-1-oxa-8-azaspiro[4.5]decane
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
2-{1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)-N-(4-methoxy-2-methylphenyl)propanamide
4-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(1-methyl-1H-pyrazol-3-yl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-4-oxo-2-propyl-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
3-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-1-(4-methylphenyl)urea
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-oxo-3,4-dihydroquinazoline-2-carboxamide
(3aS,6aS)-5-(4-methylphthalazin-1-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(thiomorpholin-4-yl)butan-1-one
5-[2-(morpholin-4-ylmethyl)phenyl]pyridine-2-carbonitrile
4-{2-[3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}phenol