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{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-(2-methoxyethyl)-9-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{1-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}pyridine
2-cyclopropyl-1-[4-(1H-pyrazol-4-yl)phenyl]-1H-imidazole
4-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
5-(cyclopropylmethyl)-3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}pyrrolidin-3-yl)-N-methylacetamide
4-{4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-[2-methyl-2-(morpholin-4-yl)propyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-cyclohexyl-1-(2-hydroxyethyl)-N-(pyridin-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-(3-methoxyphenyl)pyrrolidin-3-yl]-2-(propan-2-yloxy)acetamide
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-(butan-2-yl)-N-[(3-chlorophenyl)methyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(trifluoromethyl)piperidine
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-2,4-dimethylpyridine
8-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{2-[4-(1H-1,3-benzodiazol-2-ylmethyl)morpholin-2-yl]ethyl}-2,2-dimethylpropanamide
4-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-1λ6-thiomorpholine-1,1-dione
{[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
4-methanesulfonyl-2-{[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]formamido}butanoic acid
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-[4-(6,8-dimethylquinolin-4-yl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
6-[3-(hydroxymethyl)pyrrolidin-1-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
(3R,7S,8aS)-3-methyl-7-{[(4-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(4-chloro-1-methyl-1H-indole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
5-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(4-propanoylphenoxy)acetamide
1-{1-[1-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-2-ethylpyrimidine-5-carboxamide
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-3,4-dimethoxybenzamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine
(3S,4S)-4-(dimethylamino)-1-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
N-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
ethyl 4-({1-[4-(dimethylcarbamoyl)phenyl]piperidin-4-yl}amino)piperidine-1-carboxylate
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3-phenylprop-2-ynoyl)piperidine-4-carboxamide
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-(propan-2-yl)pyrimidin-2-amine
4-(1H-pyrazol-3-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}benzamide
2-{[6-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)pyridazin-3-yl](methyl)amino}ethan-1-ol
(2R,6S)-2,6-dimethyl-4-[2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]morpholine
1-[2-(propan-2-ylsulfanyl)ethyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-[(2,4-dichlorophenyl)methyl]-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{4-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]morpholin-3-yl}acetic acid
5-[3-oxo-3-(3-phenylpiperidin-1-yl)propyl]-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
methyl 2-({5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-yl}formamido)acetate
3-{6-[ethyl(methyl)amino]pyrimidin-4-yl}-5-[2-(piperidin-2-yl)ethyl]phenol
7-(cyclobutylmethyl)-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-aminoethyl)-N-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,3-triazole-4-carboxamide