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3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
1-(3-ethoxyphenyl)-3-[1-(morpholine-4-carbonyl)piperidin-4-yl]urea
(4aS,8aS)-2-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
2-{4-[5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenyl}pyridine
1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
1-methyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4S)-4-amino-1-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
[7-(5-fluoropyridin-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-(furan-2-ylmethyl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-4-carboxamide
methyl 2-(diethylsulfamoyl)-6-[(2,4-difluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]ethan-1-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
4-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3,5-dimethyl-1H-pyrazole
{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
2-{1-[1-(2-methylquinolin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
6-methyl-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-methyl-N-[2-(phenylsulfanyl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-N,N-dimethylazepan-4-amine
2-(dimethylamino)-1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
N-{[(2S,4S)-4-fluoro-1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}pyrrolidin-2-yl]methyl}pentanamide
(3R,4S)-1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-4-phenylpyrrolidin-3-amine
6-[methyl(thiophen-3-ylmethyl)amino]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
3-{[2-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
(2S,4S)-4-cyclobutaneamido-N-ethyl-1-(1H-indol-5-ylmethyl)pyrrolidine-2-carboxamide
8-[4-(4-fluorophenyl)oxane-4-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[(4-methylphenyl)methyl]-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
2-ethoxy-5-(2-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrimidin-4-yl)benzoic acid
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}cyclopentane-1,3-dicarboxamide
1-(carbamoylmethyl)-N-(2-methylbut-3-yn-2-yl)piperidine-3-carboxamide
2-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(naphthalen-1-ylmethyl)-4-[(pyridin-3-ylmethyl)amino]pyrrolidin-2-one
4-{[2-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
3-{[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]methyl}-1λ6-thiolane-1,1-dione
2-{[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl](propan-2-yl)amino}ethan-1-ol
1-benzyl-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
2-ethyl-N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
N-tert-butyl-2-{[1-(1H-imidazol-1-yl)propan-2-yl]amino}acetamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
(8aS)-2-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
3-chloro-4-{[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
(1R,7S)-N-cyclopropyl-3-(2-ethylbutyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-(4-fluoro-2-methylphenoxy)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidine-4-carboxylic acid
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(3-methoxyphenoxy)ethan-1-one
4-(1H-pyrazol-3-yl)-N-[2-(pyridin-4-yl)ethyl]benzamide
4-hydroxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(7S,9aR)-N-cyclohexyl-7-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-(3-phenylpiperidin-1-yl)acetamide