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3-(3,4-dimethoxybenzoyl)-1-(1,4-dithiepan-6-yl)piperidine
(2S)-2-(6-ethyl-4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
1-(4-hydroxybenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-[1-(azepan-1-yl)-1-oxopropan-2-yl]-1-(2-methoxyphenyl)piperazin-2-one
6-fluoro-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-ethyl-5-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}pyrimidin-2-amine
3-[ethyl({[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
5-[1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
N-[2-(furan-2-yl)ethyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
9-(2-methoxyethyl)-1-methyl-4-[2-(2-oxopyrrolidin-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-(2,5-dimethylphenyl)-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
N,N-dimethyl-2-[methyl({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amino]propanamide
2-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
(2S,4S)-1-benzyl-N-[2-(2-fluorophenyl)ethyl]-4-[(1-methylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
{[4-(methylsulfanyl)phenyl]methyl}(propyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
1-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1,2-oxazol-5-yl}methyl)-2-methyl-1H-1,3-benzodiazole
N-cyclopentyl-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
(3R)-3,4,4-trimethyl-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]pyrrolidin-3-ol
N-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2,5-dioxoimidazolidin-4-yl)acetamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-5-(4-methoxyphenyl)furan-2-carboxamide
3-{[(4,6-dimethylpyridin-3-yl)methyl]sulfamoyl}-N-(2-methoxyethyl)benzamide
3-{4-phenyl-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}propan-1-ol
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
3-cyclopropyl-5-[2-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)ethyl]-1H-1,2,4-triazole
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]butan-1-one
3-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}benzonitrile
1-[(4-ethylphenyl)methyl]-4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}pyrrolidin-2-one
5-(4-methanesulfonylpiperazine-1-carbonyl)-N,N,4-trimethylpyrimidin-2-amine
7-methyl-4-(2-methylpyrrolidine-1-carbonyl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline
N-{4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}acetamide
5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
4-[(1-cyclobutanecarbonylpiperidin-4-yl)oxy]-N-(2-phenylethyl)benzamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrazol-1-yl]acetamide
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
(3S)-3-ethyl-4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]morpholine
ethyl 2-{1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperidin-2-yl}acetate
6,7-dimethoxy-2-(5-methylpyridin-3-yl)quinazolin-4-amine
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(1,3-dihydroxypropan-2-yl)piperidine-3-carboxamide
5-cyclopropyl-N-(2-methoxyethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}thieno[2,3-d]pyrimidine-6-carboxamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1,3-benzothiazole-6-carboxamide
5-{[2-(4-chlorophenyl)ethyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 2-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-1,3-oxazole-4-carboxylate
3-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
2-(3-methyl-1,2-oxazol-5-yl)-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxylic acid