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3-[(3R,4S)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
1-[(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
4-[methyl({3-[(4-methylphenyl)sulfanyl]propyl})amino]pyrimidine-5-carboxylic acid
(2S,4S)-4-acetamido-N,N-diethyl-1-[(5-fluoro-2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-3-phenyl-1H-pyrazole-4-carboxamide
N-[(1R)-1-(3-methoxyphenyl)ethyl]-3-azaspiro[5.5]undecan-9-amine
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
3-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
1-(2-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-[2-(3-fluorophenyl)-2-hydroxyethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-{4-[(propylamino)methyl]phenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3,6-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
1-[(4-fluorophenyl)methyl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
3-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1-[4-(1H-pyrazol-5-yl)phenyl]urea
methyl 3-[(3S,4R)-1-{[4-(diethylamino)-2-hydroxyphenyl]methyl}-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
1-{3-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-5-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
(7R,9aR)-N-benzyl-7-[(benzylsulfanyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
(2S,4S,5R)-5-(2-chlorophenyl)-4-[4-(hydroxymethyl)piperidine-1-carbonyl]-1,2-dimethylpyrrolidine-2-carboxylic acid
2-[(2-{1-[4-(propan-2-yl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
5-{[(4-chlorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}acetate
4-(benzyloxy)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine
4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-[4-(propan-2-yl)phenyl]-1H-pyrazole
2-benzyl-8-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-hydroxy-N-(1-phenylbutyl)benzamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]acetamide
(1S,5R)-3-(3-ethoxypropanoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-fluorophenyl)-3-{1-[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
methyl 5-(quinolin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-[(thian-4-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
2-{[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
4-(4-cyclopropanecarbonylphenyl)-N,N-diethylbenzamide
(3S,4R)-1-[2-(furan-2-yl)-2-oxoacetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-{2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}pyrrolidin-2-one
(2S)-1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidine-2-carboxamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-5-ylmethyl)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-methyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
1-(4-{[3-(2-phenylpyridin-4-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
(1R,5S,6S)-6-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-1,4-diazepan-5-one
3-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[(3-methoxyphenyl)methyl]-3-[1-(8-methoxyquinolin-2-yl)piperidin-3-yl]propanamide
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl}){[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-(5-{1-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
4-{2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxoethyl}piperazin-2-one