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N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pent-4-enamide
7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-[6-(piperidin-1-yl)pyridin-3-yl]-2-(thiomorpholin-4-yl)acetic acid
5-chloro-4-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1,3-dimethyl-1H-pyrazole
N-phenyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-(3-cyclohexyl-1H-pyrazol-4-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
3-(1-benzyl-1H-imidazol-2-yl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
(1R,5S,8R)-3-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
1-methyl-4-(5-methyl-2-phenylfuran-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-cyclopentyl-N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
1'-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
5-chloro-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]thiophene-2-carboxamide
1-(furan-2-carbonyl)-4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-1,4-diazepane
4-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}benzoic acid
8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(3-methylbut-2-en-1-yl)-8-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[1-(1H-indol-5-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
2-(2-methoxyphenoxy)-N-{[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}acetamide
(dicyclopropylmethyl)(methyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
2-{[1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxy}-1,3-benzothiazole
5-(oxolan-2-ylmethyl)-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(2-fluoro-3-methylphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N4,N4,5-trimethyl-N2-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidine-2,4-diamine
3-(1-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)phenol
4-(4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
4,6-dimethyl-1-(2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
1-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-ol
3-(3-cyclopropyl-5-{[(2-ethyl-6-methylpyridin-3-yl)oxy]methyl}-1H-1,2,4-triazol-1-yl)-1λ6-thiolane-1,1-dione
1-{2-amino-4-[(cyclopent-3-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-ethoxyethan-1-one
2-(3-acetyl-1H-indol-1-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]acetamide
2-methyl-4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine
4-[1-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)ethyl]morpholine
N-(dimethyl-1,2-oxazol-4-yl)-4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
2-(methylsulfanyl)-5-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)pyrimidine
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-butyl-5-methoxy-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(pyridin-3-ylmethyl)acetamide
3-(3-methoxyphenyl)-4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
3-(1-benzyl-1H-imidazol-2-yl)-1-(5-methylthiophene-3-carbonyl)piperidine
2-amino-7-[4-(1H-pyrazol-3-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-benzyl-4-(1-benzyl-1H-pyrazole-4-carbonyl)piperazin-2-one
(2S)-2-hydroxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}propanamide
3-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-[3-(sulfamoylmethyl)phenyl]urea
methyl 3-cyclohexyl-1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
7-[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
2-(2,3-dimethoxy-5-methylphenyl)-2-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]acetic acid