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2-[1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
3-methoxy-N-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]piperidine-1-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(ethylamino)-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)pyrimidine-5-carboxamide
2-[(1S,5R)-3-(2-methoxypyridine-4-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-{2-[1-(propan-2-yl)piperidine-4-carbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
(3S)-3-ethyl-4-[(1-methyl-1H-imidazol-4-yl)sulfonyl]morpholine
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-ethyl-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(5-methyl-1H-pyrazol-1-yl)acetamide
1-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]pyrimidine
(2R)-N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}oxolane-2-carboxamide
2-methyl-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-ethyl-2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-methylpyrimidine
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-N-(1-methyl-1H-1,2,4-triazol-3-yl)benzamide
2-({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-(3-methoxypropyl)-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
7-methoxy-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[2-(pyridin-2-yl)ethyl]quinoline-4-carboxamide
2-{[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
N-methyl-N-[2-(pyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(2-phenylpropyl)-1H-1,2,3-triazole
ethyl 4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-[({[1-(2-hydroxyethyl)piperidin-4-yl]methyl}(methyl)amino)methyl]-6-methylquinolin-4-ol
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-(2-phenylethyl)propanamide
N,N-dimethyl-2-[(1,2,3,4-tetrahydronaphthalen-2-ylformamido)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
6-[1-(1-benzoxepine-4-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-(3-ethylphenyl)-5-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[3-(pyridin-2-yl)propyl]-6-(quinolin-3-yl)pyridine-3-carboxamide
N5-cyclopropyl-N6-[2-(6-methylpyridin-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
2-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-6-(4-fluorophenyl)pyridine-3-carboxylic acid
[(2-butoxy-3-methoxyphenyl)methyl][1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amine
5-ethoxy-N-(isoquinolin-5-ylmethyl)-N-methylfuran-2-carboxamide
N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
(2E)-N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(thiophen-2-yl)prop-2-enamide
(2S,4R)-1-benzyl-4-{[(2,6-difluorophenyl)methyl]amino}-N,N-diethylpyrrolidine-2-carboxamide
(1S,5R)-3-benzyl-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(4-fluorophenyl)piperidin-4-ol
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
[(3aS,6aS)-2-(trimethylpyrimidin-4-yl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane