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(cyclopentylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
(4aS,7aR)-1-(3,4-difluorobenzoyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1H-imidazol-1-yl)-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}butan-1-one
4-[(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-2-yl)methyl]morpholine
(2S,4R)-4-amino-N-methyl-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidine-2-carboxamide
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
5-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
5-methyl-N-[4-(pyridin-2-yl)butyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2R,6S)-2,6-dimethyl-4-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}morpholine
1-(1,2,3,4-tetrahydroisoquinolin-2-yl)-3-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)propan-1-one
2-methyl-6-{4-[(propan-2-yloxy)methyl]piperidine-1-carbonyl}-4H-pyran-4-one
4-(cyclopropylmethyl)-1-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-[({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)amino]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-4-(2-oxopyrrolidin-1-yl)butanamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-methyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-2-methoxypyrimidine
(2S,4R)-4-(dimethylamino)-1-(2-hydroxynaphthalene-1-carbonyl)pyrrolidine-2-carboxylic acid
6-methyl-N4-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrimidine-2,4-diamine
N-{1-[2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)acetyl]pyrrolidin-3-yl}-N-methylacetamide
(1S,5R)-6-(3-phenoxypropyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(thiophen-3-yl)propan-1-one
1-ethyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1-ethyl-1H-indazol-3-yl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(4-fluorophenyl)methyl]-2-[methyl(piperidin-4-yl)amino]-N-(pyridin-4-ylmethyl)acetamide
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-4-phenoxybutan-1-one
[(2-ethoxypyridin-3-yl)methyl]({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl})amine
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methoxyethan-1-one
2-{2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
N,N-diethyl-1-[1-(quinolin-7-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-{[5-(2,5-dimethoxyphenyl)-2-hydroxyphenyl]methyl}piperidine-3-carboxamide
1-[2-({[(2,4-difluorophenyl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-[4-methyl-2-({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amino)pyrimidin-5-yl]ethan-1-one
2-({[(3R,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
1-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]piperidin-4-ol
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
3-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidin-2-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-2-(thiophen-2-ylformamido)propanamide
N-(3-methylphenyl)-4-[(oxolan-3-yl)sulfamoyl]benzamide
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-(piperidine-1-carbonyl)piperidine
N-benzyl-N-ethyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
6-{1-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}-2-phenyl-3,4-dihydropyrimidin-4-one
8-[(4-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-oxo-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
[2-(diethylamino)ethyl]({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
1-[2-(3-chlorophenyl)ethyl]-4-{[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amino}pyrrolidin-2-one
5-benzamido-1-cyclopentyl-N-[2-(1H-imidazol-1-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide