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[1-(3-{[6-(propan-2-yl)pyrimidin-4-yl]amino}propyl)piperidin-3-yl]methanol
5,7-dimethyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}urea
5-(2-fluorophenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{1'-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
2,3,5-trimethyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(3-ethoxypropyl)-1H-pyrazole-4-carboxamide
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-6-methoxyphenol
methyl 2-[4-(pyridin-3-yl)piperazine-1-carbonyl]piperidine-1-carboxylate
5-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]pyridine-2-carbonitrile
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-3-(4-methoxyphenyl)propan-1-one
[1-({[(2E)-3-(furan-2-yl)prop-2-en-1-yl](methyl)amino}methyl)cyclopentyl]methanol
1-ethyl-N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
N-[1-(pyrazin-2-yl)propan-2-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}benzonitrile
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-(pyridin-2-yl)propan-1-one
N-[2-(furan-2-yl)ethyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
(3S,9aR)-3-(2-methylpropyl)-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-amino-3-ethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
N-{2-[(4-chloro-1H-pyrrol-2-yl)formamido]ethyl}pyridine-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-phenyl-1,2-oxazole-5-carboxamide
(2S,3S)-2-{[4-hydroxy-2-(3-methylphenyl)pyrimidin-5-yl]formamido}-3-methylpentanamide
4-({1-[(4-fluorophenyl)methyl]-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
1-(4-chlorophenyl)-N-{[1-(1,4-dithiepan-6-yl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-methyl-4-[3-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-methyl-N-(pyridin-2-ylmethyl)piperidin-4-amine
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]methyl}piperidin-2-one
1-(4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-{2-chloro-4-[1-(pyridin-3-yl)-1H-imidazol-2-yl]phenoxy}acetamide
methyl(oxolan-3-ylmethyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
N-cyclopropyl-2,3-dimethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-indole-7-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pyridin-3-ylmethyl)pyridine-3-carboxamide
4-benzyl-3-{2-[4-(2-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
7-chloro-2-{[(dimethylsulfamoyl)amino]methyl}-N-[(4-fluorophenyl)methyl]quinazolin-4-amine
5-chloro-1,3-dimethyl-4-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
3-[methyl({[1-propyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
3-({[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]carbamoyl}amino)-N-ethylbenzamide
3-(3-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine-2-carbonitrile
3-[(3R,4S)-4-(dimethylamino)-1-[2-(3-methoxyphenyl)acetyl]piperidin-3-yl]propanoic acid
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2,4-difluorophenyl)methyl]methylamine
[2-(1H-imidazol-4-yl)ethyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-[1-(4-cyclopropanecarbonylphenyl)-1H-pyrazol-3-yl]pyrazine