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(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(2,2,2-trifluoroethyl)carbamoyl]pyrrolidine-2-carboxylic acid
ethyl 1-(2-hydroxyethyl)-5-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-2-(morpholin-3-yl)acetamide
(4aR,7aS)-1-acetyl-4-(2-chlorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1'-(3-methoxypyrazin-2-yl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-[2-(3-chlorophenyl)ethyl]-2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]acetamide
5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-1H-indole
1-(2,2-diphenylacetyl)-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
N-[(4-hydroxyphenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
{[2-(4-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}(2-methoxyethyl)methylamine
N-(oxan-4-yl)-5-(oxolan-2-yl)thiophene-2-carboxamide
N-(cyclopropylmethyl)-N-(2-methoxyethyl)-4-methyl-3-phenyl-1H-pyrazole-5-carboxamide
2-cyclopentyl-N-cyclopropyl-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)acetamide
N,N-bis(2-hydroxyethyl)-5-methyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
dimethyl(1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]phenyl}ethyl)amine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}acetamide
N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
1-[2-hydroxy-3-(3-{1-oxa-7-azaspiro[3.5]nonan-7-ylmethyl}phenoxy)propyl]piperidin-4-ol
1-[(3-chlorophenyl)methyl]-4-[2-(pyrrolidin-1-yl)benzoyl]piperazine
N-[1-(cyclohex-1-en-1-yl)ethyl]-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)piperazine
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-methylacetamide
2-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-2-methylimidazo[1,2-a]pyridine-6-carboxamide
1-[(3-methoxyphenyl)methyl]-4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazin-2-one
1-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-methoxyethan-1-one
5-methyl-2-phenyl-4-{3-propyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-imidazole
{[2-(azocan-1-yl)pyridin-3-yl]methyl}({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})amine
6-[1-(2,5-difluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
4,5-dimethyl-6-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}pyrimidin-2-amine
4-benzyl-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3-ethyl-1,4-diazepan-5-one
5-[(3-fluorophenyl)methyl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
2-(4-fluoro-2-methoxyphenyl)-2-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]acetic acid
3-(2-methoxyethyl)-5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazole
1-[(3-fluorophenyl)methyl]-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-6-oxopiperidine-3-carboxamide
6-chloro-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-fluoro-N-(propan-2-yl)imidazo[1,2-a]pyridine-2-carboxamide
1,3,6-trimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4S)-1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-4-propylpyrrolidine-3-carboxylic acid
N-(3-methoxyphenyl)-5-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-amine
2-{3-[2-(trifluoromethyl)morpholine-4-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
N-ethyl-5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidin-2-amine
3-ethyl-1-(5-ethyl-1,3,4-thiadiazol-2-yl)piperidine-3-carboxylic acid
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-amino-6-(4-fluorophenyl)-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
4-cyclobutaneamido-N-[2-(methylsulfamoyl)ethyl]benzamide
N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
2-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-N-methylpyridine-4-carboxamide