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5-methyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-1,2,4-oxadiazole
2-[(3-methoxyphenyl)methyl]-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)morpholine
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
5,6-dimethoxy-2-({5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-1,2-dihydroisoquinolin-1-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-[2-(dimethylamino)ethyl]-5-(furan-2-yl)-1H-pyrazole-4-carboxamide
1-(2-methoxyethyl)-N-[(4-phenylphenyl)methyl]pyrrolidine-3-carboxamide
3-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-2-ol
4-{5-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)ethyl]-1-ethyl-1H-1,2,4-triazol-3-yl}benzamide
5-amino-4-chloro-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-(pyrrolidine-1-sulfonyl)-4-(thiophen-3-ylmethyl)piperazine
1-cyclopropyl-6-oxo-N-[(3-phenoxyphenyl)methyl]piperidine-3-carboxamide
2-(3-fluorophenyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
3-cyclopropaneamido-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-methylbenzamide
1-(cyclohexylmethyl)-6-oxo-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)thiophene-2-sulfonamide
3-methyl-3-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-(2-methylquinolin-8-yl)urea
N-[(5-methylpyrazin-2-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
N-[(4,6-dimethylpyridin-3-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[(2S,4R)-1-[(3-fluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
9-(2-methyl-6-propylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrimidin-4-amine
2-[2-(2-phenylethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
7-propyl-2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,7-diazaspiro[4.5]decan-6-one
1'-[(3-chloropyridin-4-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
methyl (2S,4R)-4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}pyrrolidine-2-carboxylate
N-{4-[2-(dimethylamino)ethoxy]-1-(3-fluorophenyl)-1H-indazol-3-yl}pyridazine-3-carboxamide
N-[(4,6-dimethylpyridin-3-yl)methyl]-2-methyl-6-(propan-2-yl)pyrimidin-4-amine
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(morpholin-3-yl)ethan-1-one
2-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1-benzofuran-5-carboxamide
3-chloro-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
3-[(1-acetylpiperidin-3-yl)methyl]-6-ethyl-5-phenyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
8-[2-(ethylsulfanyl)propanoyl]-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1'-(5-chloro-2-fluorobenzoyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-(4-fluorophenyl)-N,3,5-trimethyl-1H-pyrazole-4-carboxamide
N-[2-(furan-2-yl)ethyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
6-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-2,3-dimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
4-[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]-2-methoxyphenol
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(thiophen-2-yl)propan-1-one
2-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-phenyl-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]morpholine
(2S,4R)-4-(cycloheptylamino)-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
5-[2-(5-methylfuran-2-yl)propyl]-4-phenyl-1H-imidazole
(4aS,7aR)-1-[(4-hydroxy-3-methylphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(1,3-thiazole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
4-(2-phenylbenzoyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
2-[3-(pyrrolidin-1-yl)pyrazin-2-yl]benzoic acid