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N'-[2-(methylsulfanyl)phenyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]butanediamide
4-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}pyridine
2-(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-3-yl)-1,3-benzoxazole
1-({4-[1-(3-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]phenyl}methyl)-4-methylpiperazine
[(3R,4R)-1-(2,3-dimethyl-1H-indole-7-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-8-methyl-1,2-dihydroquinolin-2-one
5-[1-(cyclopropylmethyl)pyrrolidin-2-yl]-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]thiophene-2-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
3-{1-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
2-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-1,2-dihydroisoquinolin-1-one
2,5-dimethyl-4-(3-{1-[(6-methylpyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
N-ethyl-N-[2-(4-methoxyphenoxy)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-ethyl-N-methylpyridine-3-carboxamide
2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-8-methoxyquinoline
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(1,3-thiazol-2-ylmethyl)amine
1-(2-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}pyrimidin-4-yl)piperidin-4-ol
(2S,4R)-4-amino-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
1-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
3-(1-{[7-(methylsulfanyl)-2-oxo-1,2-dihydroquinolin-3-yl]methyl}piperidin-3-yl)propanamide
1-(cyclopropylmethyl)-5-(3-fluoro-4-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[4-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)phenyl]ethan-1-one
ethyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-phenylpyridazin-3-amine
N-[2-(dimethylamino)ethyl]-4-(quinolin-6-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-cyclohexyl-N-[(4-fluorophenyl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
4-(naphthalen-1-ylmethyl)-3-{2-oxo-2-[4-(piperidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
5-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(cyclobutylmethyl)piperazine-1-carbonyl]isoquinoline
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
1-ethyl-5-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1H-1,2,4-triazole
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]propan-1-one
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
1-[3-(cyclohexylsulfanyl)propyl]-3-(1,3-dimethyl-1H-pyrazol-4-yl)urea
3-[3-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-{4-[(5-acetylthiophen-3-yl)methyl]morpholin-3-yl}-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
1-[(2-fluorophenyl)methyl]-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[3-methoxy-5-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
2-chloro-N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-acetamido-N-methylbenzamide
2-(3-hydroxypropyl)-9-{[2-(methylsulfanyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-phenyl-1-(1,3,7-trimethyl-1H-indole-2-carbonyl)piperidin-3-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,3-oxazole-4-carboxamide
1-(cyclohexylmethyl)-3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
2-(2-butoxy-4-fluorophenyl)-3-(pyrrolidine-1-carbonyl)pyridine
3-(1H-1,3-benzodiazol-2-ylmethyl)-6-(4-fluorophenyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one