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4-[4-(4-cyclohexylphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
3-{1-[(2-amino-5-ethylpyrimidin-4-yl)amino]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
N-(1H-imidazol-2-ylmethyl)-N,2-dimethyl-5-propylpyrimidin-4-amine
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
(1R,3S,5S)-3-(4-methoxyphenyl)-8-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-8-azabicyclo[3.2.1]octane
2-(4-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-[3-(methylamino)propyl]-3-(5-methylfuran-2-yl)benzamide
2-(2-chlorophenyl)-1-[3-(4-fluorophenoxy)azetidin-1-yl]-2-hydroxyethan-1-one
1'-(5-ethyl-1,2-oxazole-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
[(2S,4R)-4-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]-1-methylpyrrolidin-2-yl]methanol
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
(1S,5R)-6-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
5-{[(2,3-difluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(3-methoxypropyl)benzamide
N-[3-(dimethylamino)propyl]-5-methyl-6-(morpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine
4-(2-fluoro-4,5-dimethoxyphenyl)-1-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl N-({methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]carbamoyl}methyl)carbamate
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dimethylquinoxaline-6-carboxamide
8-[(4-hydroxyphenyl)methyl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
(1R,5R)-6-[3-(4-fluorophenoxy)propyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
(1H-1,3-benzodiazol-2-ylmethyl)(methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
2-(5-methyl-1H-pyrazol-1-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
5-{2-[(naphthalen-2-ylmethyl)amino]ethyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]pyrrolidin-2-one
2-(2-methyl-1,3-thiazol-4-yl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-[4-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)thiophen-2-yl]ethan-1-one
2-(3-hydroxypropyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2,6-dimethylquinoline-4-carboxamide
2-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-1,2-oxazolidin-4-ol
2-[7-(1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-ol
(4S)-1-[(1-ethyl-1H-pyrazol-3-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
6-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-5-methyl-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
3-[4-(5-acetylpyridin-2-yl)piperazin-1-yl]propanamide
5-[2-(4-chlorophenyl)morpholine-4-carbonyl]quinoxaline
4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazin-2-one
2-({[(3-chlorophenyl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
{4-[(2-aminopyridin-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-(2,2-diphenylethyl)-4-(5-methyl-1,2-oxazole-3-carbonyl)morpholine
(1S,5R)-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-hydroxycyclohexyl)methyl]-5-methyl-2-phenylfuran-3-carboxamide
2-(2-methoxyethyl)-8-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one