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5-{2-[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]ethyl}-1,3,4-thiadiazol-2-amine
[(5-fluoro-3-methyl-1H-indol-2-yl)methyl](methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
2-{1-[(3,4-difluorophenyl)methyl]-4-(1H-indol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-cyclopropyl-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1,2,3,4-tetrahydroquinoline-8-carboxamide
3-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]benzamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(2,5-dimethoxybenzenesulfonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
11-{[(3,5-difluorophenyl)methyl]amino}-4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine-1-carboxamide
N-[(3S,4R)-1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-(2-hydroxyphenyl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H-pyrazole-5-carboxamide
7-(5-chloropyridin-2-yl)-4-[2-(1H-pyrazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4R)-4-amino-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
N2-(2-methoxyethyl)-N4-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
methyl 4-{[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}thiophene-2-carboxylate
4,6-dihydroxy-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyridine-3-carboxamide
4-(4-methylpiperazin-1-yl)-N-(1-phenylbutyl)benzamide
(2S,4S)-4-[4-(4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}phenyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]urea
(2R)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]pyrrolidine-2-carboxamide
2-methyl-5-{4-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N,N-dimethyl-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)thiophene-2-carboxamide
2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-1-(piperidin-1-yl)propan-1-one
N-methyl-N-(quinolin-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-(4-chloro-1H-indazol-1-yl)-N-(2-propyl-2H-1,2,3-triazol-4-yl)acetamide
N-(cyclohexylmethyl)-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
ethyl 4-{3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}piperidine-1-carboxylate
(3S,7S)-5-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
5-{[1-(2-methoxyphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(2-fluorophenyl)ethyl]acetamide
3-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-N-(furan-2-ylmethyl)propanamide
3-{2-[4-(2-methanesulfonylethyl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
1-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
1-cyclopentyl-5-(2-methylpiperidine-1-carbonyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(piperidin-1-yl)ethyl]amine
2-{[2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
2-benzyl-5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
N-(cyclohexylmethyl)-4-oxo-1-(propan-2-yl)-5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
3-cyclopropyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
(3R)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
6-methyl-3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(1-benzylpiperidin-4-yl)-N-(2-hydroxyethyl)-N-methylpiperidine-3-carboxamide
8-{[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]methyl}-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-2-one
1-{3-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}azepan-2-one